Tehran University of Medical Sciences
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Alireza Foroumadi

Contact Information
Tel: 02166954708
Fax: 02166461178
Address: Faculty of Pharmacy and Pharmaceutical Sciences Research Center, Tehran University of Medical Sciences, Tehran, Iran.
Academic Rank
Professor
School
Pharmacy
Medicinal Chemistry
Research Center
Pharmaceutical Sciences Research Center
About
CV last edited on: 2019/16/01

1.

Fellowship


Postdoctoral Research Fellow, School of Pharmaceutical Sciences, Teikyo University, Tokyo, Japan, Aug 1996–Feb 1997
Supervisor: Prof. S. Ikegami
2.

Fellowship


Postdoctoral Research Fellow, School of Pharmaceutical Sciences, University College London, London, UK , Sep 2002–Feb 2003
Supervisor:Prof. C. R. Ganellin
3.

Pharm D


Doctorate of Pharmacy (Pharm.D.) , Tehran University of Medical Sciences, tehran, iran, 1990
4.

Ph.D


Ph.D. in Medicinal Chemistry, Tehran University of Medical Sciences, tehran, iran, 1996

Scientific Position

1.

Professor, Pharmaceutical Sciences Research Center


Tehran University of Medical Sciences, Dec 2007-present
2.

Associate Professor, Pharmaceutical Sciences Research Center


Tehran University of Medical Sciences, 2005 -2007
3.

Associate Professor , Faculty of Pharmacy


Kerman University of Medical Sciences, June 2002- 2004
4.

Assistant Professor, Faculty of Pharmacy


Kerman University of Medical Sciences, 1996 -2002

English

1.

Hydrobromic Acid


Authors: A Foroumadi and M Saeedi
English , Publisher: Elsevier Inc, 2014, Original
2.

2-Mercaptoethanol


Authors: A Foroumadi and M Saeedi
English , Publisher: Elsevier Inc , 2014, Original

English

1.

Glycidol


Authors: A Foroumadi, S Emami
English, Publisher: Elsevier Inc, 2014, Original

Farsi

1.

An Introduction to Practical Organic Chemistry, Vol. 1


Authors: Foroumadi A., Yazdanian M
Farsi, Publisher: Teymoorzadeh Publication Co, Original

Papers

English

1.

A one-pot, three-component, solvent-free synthesis of novel 6h-chromeno[3’,4’:5,6]pyrido[2,3-d]pyrimidine-triones under microwave irradiation


Authors: Firoozpour L, Yahyavi H, Ejtemaei R, Moghimi S, Foroumadi A*
Journal of Chemical Research, Vol.42, No.12, Year. 2018,
2.

Spectroscopic and molecular docking studies on DNA binding interaction of podophyllotoxin


Authors: Heidary Alizadeh B, Dehghan Gh, Derakhsh Ahmadi V, Moghimi S, Asadipour A, Foroumadi A
Journal of Sciences, Islamic Republic of Iran, Vol.29, No.2, Year. 2018,
3.

N-substituted piperazinyl sarafloxacin derivatives: synthesis and in vitro antibacterial evaluation


Authors: Asadipour A, Moshafi M.H, Khosravani L, Moghimi S, Amou E, Firoozpour L, Ilbeigi G, Beiki K, Soleimani E, Foroumadi A*
DARU, Journal of Pharmaceutical Sciences, Vol.26, No.2, Year. 2018,
4.

New 7-piperazinylquinolones containing (benzo[d]imidazol-2-yl)methyl moiety as potent antibacterial agents


Authors: Arab H, Faramarzi M, Samadi N, Irannejad H, Foroumadi A, Emami S
Molecular Diversity, Vol.22, No.4, Year. 2018,
5.

Synthesis and cholinesterase inhibitory activity of new 2-benzofuran carboxamide-benzylpyridinum salts


Authors: Abedinifar F, Farnia S, Mahdavi M, Nadri H, Moradi A, Ghasemi J, Küçükkılınç T.T, Firoozpour L, Foroumadi A*
Bioorganic Chemistry , Vol.80, Year. 2018,
6.

Synthesis and biological evaluation of 2-phenyl benzothiazole derivatives as cytotoxic agents


Authors: Firoozpour L, Mokhtari A, Moghimi S, Safavi M, Foroumadi, A
Journal of Chemical Sciences, Vol.29, No.4, Year. 2018,
7.

Novel 3-phenylcoumarin–lipoic acid conjugates as multi-functional agents for potential treatment of Alzheimer's disease


Authors: Jalili-Baleh L, Nadri H, Forootanfar H, Samzadeh-Kermani A, Küçükkılınç T.T, Ayazgok B, Rahimifard M, Baeeri M, Doostmohammadi M, Firoozpour L, Bukhari S, Abdollahi M, Ganjali M, Emami S, Khoobi M, Foroumadi A*
Bioorganic Chemistry, Vol.79, Year. 2018,
8.

Synthesis and biological evaluation of new coumarins bearing 2,4-diaminothiazole-5-carbonyl moiety


Authors: Ayati A, Oghabi Bakhshaiesh T, Moghimi S, Esmaeili R, Majidzadeh-A K, Safavi M, Firoozpour L, Emami S, Foroumadi A
European Journal of Medicinal Chemistry, Vol.155, No.15, Year. 2018,
9.

. Glutathione conjugated polyethylenimine on the surface of Fe3O4 magnetic nanoparticles as a theranostic agent for targeted and controlled curcumin delivery


Authors: Aeineh N, Salehi F, Akrami M, Nemati F, Alipour M, Ghorbani M, Nikfar B, Salehian F, Riyahi Alam N, Sadat Ebrahimi S, Foroumadi A*. Khoobi M, Rouini M, Dibaei M, Haririan I, Ganjali M, Safaei S
Journal of Biomaterials Science, Vol.29, No.10, Year. 2018,
10.

An eco-friendly synthesis of 4-aryl-substituted pyrano-fuzed coumarins as potential pharmacological active heterocycles using molybdenum oxide nanoparticles as an effective and recyclable catalyst


Authors: Pourshojaei Y, Jadidi M, Eskandari K, Foroumadi A, Asadipour A
Research on Chemical Intermediates, Vol.44, No.7, Year. 2018,
11.

Synthesis, evaluation, and molecular docking studies of aryl urea-triazole-based derivatives as anti-urease agents


Authors: Moghimi S, Goli-Garmroodi F, Allahyari-Devin M, Pilali H, Hassanzadeh M, Mahernia S, Mahdavi M, Firoozpour L, Amanlou M, Foroumadi A*
Archiv der Pharmazie, Vol.351, No.7, Year. 2018,
12.

Synthesis, docking study, and biological evaluation of novel umbellipherone/hymecromone derivatives as acetylcholinesterase/butyrylcholinesterase inhibitors


Authors: Moradi A, Faraji L, Nadri H, Hasanpour Z, Moghadam F, Pakseresht B, Golshani M, Moghimi S, Ramazani A, Firoozpour L, Khoobi M, Foroumadi, A*
Medicinal Chemistry Research, Vol.27, No.7, Year. 2018,
13.

review on flavonoid-based scaffolds as multi-target-directed ligands (MTDLs) for Alzheimer's disease


Authors: Jalili-Baleh L, Babaei E.b Abdpour S, Nasir Abbas Bukhari S, Foroumadi A, Ramazani A, Sharifzadeh M, Abdollahi M, Khoobi M
Eur. J. Med. Chem, Vol.152, Year. 2018,
14.

Design, synthesis and evaluation of novel multi-target-directed ligands for treatment of Alzheimer's disease based on coumarin and lipoic acid scaffolds


Authors: Jalili-Baleh L, Forootanfar H, Küçükkılınç, T.T, Nadri H, Abdolahi Z, Ameri A, Jafari M, Ayazgok B, Baeeri M, Rahimifard M, Abbas Bukhari S, Abdollahi M, Ganjali M, Emami S, Khoobi M, Foroumadi A*
Eur. J. Med. Chem, Vol.152, Year. 2018,
15.

Synthesis and biological evaluation of chalcone-triazole hybrid derivatives as 15-LOX inhibitors


Authors: Asadipour A, Noushini S, Moghimi S, Mahdavi M, Nadri H, Moradi A, Shabani S, Firoozpour L, Foroumadi A*
Journal of Chemical Sciences, Vol.73, No.2, Year. 2018,
16.

Synthesis and biological evaluation of 4-amino-5-cinnamoylthiazoles as chalcone-like anticancer agents


Authors: Ayati A, Esmaeili R, Moghimi S, Oghabi Bakhshaiesh T, Eslami-S Z, Majidzadeh-A K, Safavi M, Emami S, Foroumadi A*
European Journal of Medicinal Chemistry, Vol.145, Year. 2018,
17.

Caspase-dependent apoptosis induced by two synthetic halogenated flavanones, 3′,7-dichloroflavanone and 3′,6-dichloroflavanone, on human breast and prostate cancer cells


Authors: Safavi M, Shakeri R, Ardestani S, Davoodi J, Ajdary S, Foroumadi A
Biology – Animal, Vol.54, No.2, Year. 2018,
18.

Design, synthesis, cytotoxicity evaluation and docking studies of 1,2,4-triazine derivatives bearing different arylidene-hydrazinyl moieties as potential mTOR inhibitors


Authors: Ranjbar S, Edraki N, Khoshneviszadeh M, Foroumadi A*, Miri R, Khoshneviszadeh M
Research in Pharmaceutical SciencesOpen Access, Vol.13, No.1, Year. 2018,
19.

Iodine-catalyzed tandem oxidative coupling reaction: A one-pot strategy for the synthesis of new coumarin-fused pyrroles(Article)


Authors: Yahyavi H, Heravi M, Mahdavi M, Foroumadi A
etrahedron Letters, Vol.59, No.2, Year. 2018,
21.

A convenient method for the synthesis of chromeno[4,3-b]pyridines via three-component reaction


Authors: Nikookar H, Moghimi S, Sayahi M, Mahdavi M, Ranjbar P, Firoozpour, L, Foroumadi A*
Combinatorial Chemistry and High Throughput Screening48., Vol.21, No.5, Year. 2018,
22.

Design, synthesis and characterization of novel urolithin derivatives as cholinesterase inhibitor agents


Authors: Norouzbahari M, Burgaz E, Ercetin T, Fallah A, Foroumadi A, Firoozpour L, Sahin M, Gazi M, Gulcan H
Letters in Drug Design and Discovery, Vol.15, No.11, Year. 2018,
23.

Anticancer effects of synthetic hexahydrobenzo [g]chromen-4-one derivatives on human breast cancer cell lines


Authors: Pordeli M, Nakhjiri M, Safavi M, Ardestani SK, Foroumadi A
Breast Cancer, Vol.24, Year. 2017,
24.

New racemic annulated pyrazolo[1,2-b]phthalazines as tacrine-like AChE inhibitors with potential use in Alzheimer's disease


Authors: Jalili-Baleh L, Nadri H, Moradi A, Bukhari SNA, Shakibaie M, Jafari M, Golshani M, Homayouni Moghadam F, Firoozpour L, Asadipour A, Emami S, Khoobi M, Foroumadi A
Eur. J. Med. Chem, Year. 2017,
25.

An efficient approach to the synthesis of coumarin-fused dihydropyridinones


Authors: Firoozpour L, Nikookar H, Moghimi S, Mahdavi M, Asadipour A, Rashidi P, Foroumadi A
Heterocycl. Commun, Vol.23, Year. 2017,
26.

A, Synthesis and leishmanicidal activity of 1-[5-(5-nitrofuran-2-yl)-1, 3, 4-thiadiazole-2-yl]-4-benzoylepiperazines


Authors: Foroumadi A, Adibi H, Kabudanian Ardestani S, Shirooie S , Bozorgomid A, Jafari A
Iran. J. Pharm. Res, Vol.16, Year. 2017,
27.

Synthesis, cholinesterase inhibitory, and docking simulation studyIranian


Authors: Hirbod K, Jalili-Baleh L, Nadri H, Ebrahimi SES, Moradi A, Pakseresht B, Foroumadi A, Shafiee A, Khoobi M
J. Basic Med. Sciences, Vol.20, Year. 2017,
28.

Synthesis and anticholinesterase activity of new substituted benzo[d]oxazole-based derivatives


Authors: Pouramiri B, Moghimi S, Mahdavi M, Nadri H, Moradi A, Tavakolinejad-kermani E, Firoozpour L, Asadipour A, Foroumadi A
Chem. Biol. Drug Design , Vol.89, Year. 2017,
29.

Design, synthesis, molecular modeling and anticholinesterase activity of benzylidene-benzofuran-3-ones containing cyclic amine side chain


Authors: Mehrabi F, Pourshojaei Y, Moradi A, Sharifzadeh M, Khosravani L, Sabourian R, Rahmani-Nezhad S, Mohammadi-Khanaposhtani M, Mahdavi M, Asadipour A, Rahimi HR, Moghimi S, Foroumadi A
Future Med. Chem, Vol.9, Year. 2017,
30.

Synthesis and biological evaluation of novel imidazopyrimidin-3-amines as anticancer agents


Authors: Mahdavi M, Dianat S, Khavari B, Moghimi S, Abdollahi M, Safavi M, Mouradzadegun A, Kabudanian Ardestani S, Sabourian R, Emami S, Akbarzadeh T,Shafiee A, Foroumadi A
Chem. Biol. Drug Design, Vol.89, Year. 2017,
31.

An efficient four-component reaction for the synthesis of chromeno[4,3-b]quinolone derivatives


Authors: dYahya-Meymandi A, Nikookar H, Moghimi S, Mahdavi M, Firoozpour L, Asadipour A, Rashidi Ranjbar P, Foroumadi A
J. Iran. Chem. Soc, Vol.14, Year. 2017,
32.

synthetic hexahydrobenzo [g]chromen-4-one derivatives on human breast cancer cell lines


Authors: Pordeli M, Nakhjiri M, Safavi M, Ardestani SK, Foroumadi A
Breast Cancer, Year. 2017,
33.

Novel levofloxacin derivatives as potent antibacterial agents


Authors: Moshafi M. H. Bahador, N. Moghimi, S. Ejtemaei, R. A. Foroumadi A
J. Sciences, I. R. Iran, Vol.28, Year. 2017,
34.

In silico screening of IL-1β production inhibitors using chemometric toolsKhoshneviszadeh


Authors: Sakhteman A, Edraki N, Hemmateenejad B, Miri R, Foroumadi A, Shafiee A
Iran J Pharm. Res, Vol.16, Year. 2017,
35.

One-pot sequential synthesis of O-(halo-substituted benzyl) hydroxylammonium salts


Authors: Emamia S, Foroumadi A
Arab. J. Chem, Vol.10, Year. 2017,
36.

Synthesis and anti-acetylcholinesterase activity of N-[(indolyl)ethyl)- coumarin-yloxy)]alkanamides


Authors: Ghanei-Nasab S, Nadri H, Moradi A, Marjani A, Shabani Sh, Firoozpour L, Moghimi S, Khoobi M, Hadizadeh F, Foroumadi A
J. Chem. Res, Vol.41, Year. 2017,
37.

Formulation and evaluation of targeted nanoparticles for breast cancer theranostic system


Authors: Dadras P, Atyabi F, Irani S, Ma'mani L, Foroumadi A, Mirzaie ZH, Ebrahimi M, Dinarvand R
Eur. J. Pharm. Sciences, Vol.97, Year. 2017,
38.

An efficient, four-component reaction for the synthesis of novel carbamodithioates


Authors: Sadat-Ebrahimi S-E, Karim L , Moghimi S, Yahya-MeymandiA,Mahdavi M, Vosooghi M, Foroumadi A & Shafiee A
J. Sulfur Chem, Vol.38, Year. 2017,
39.

synthesis of 7-amino alkoxy homoisoflavonoides


Authors: Asadipour A, Pourshojaei Y, Eskandari K, Foroumadi A
RSC Adv, Vol.71, Year. 2017,
41.

Metal-free chemo- and regioselective acylation of pyridine derivatives with alcohols in water


Authors: Kianmehra E, Pakbazniaa A, Faghiha N, Foroumadi A
Tetrahedron, Vol.73, Year. 2017,
42.

Synthesis of Cytotoxic Isodeoxypodophyllotoxin Analogs


Authors: Alizadeh B, Emami S, Dehghan GH, Foroumadi A, Shafiee A
. J. Het. Chem, Vol.54, Year. 2017,
43.

Synthesis and cytotoxicity of novel thioxo-quinazolino[3,4-a]quinazolinones


Authors: Mohhammadhossini N, Saeedi M, Moradi S, Mahdavi M, Firuzi O, Foroumadi A, Shafiee A
Turk. J. Chem, Year. 2017,
44.

1,2,3-Triazole-isoxazole based acetylcholinesterase inhibitors: Synthesis, biological evaluation and docking study


Authors: Najafi Z, Mahdavi M, Saeedi M, Sabourian R, Khanavi M, Safavi M, Barazandeh Tehrani M, Shafiee A, Foroumadi A, Akbarzadeh T
. Lett. Drug Design Disc, Vol.14, Year. 2017,
45.

Synthesis of Novel Tacrine Analogs as Acetylcholinesterase Inhibitors


Authors: Mahdavi M, Saeedi M, Gholamnia L, Behzad Jeddi S-A, Sabourian A, Shafiee A, Foroumad A, and Tahmineh Akbarzadeh
J. Het. Chem, Vol.54, Year. 2017,
46.

Synthesis of novel benzimidazole and benzothiazole derivatives bearing a 1,2,3-triazole ring system and their acetylcholinesterase inhibitory activity


Authors: Faraji L, Shahkarami S, Nadri H, Moradi A, Saeedi M, Foroumadi A; Ramazani A; Haririan I; Ganjali M R; Shafiee A; Khoobi M
J. Chem. Res, Vol.41, Year. 2017,
47.

Facile synthesis and antiproliferative activity of 7H-benzo[7,8]chromeno[2,3-d]pyrimidin-8-amines


Authors: Akrami H, Safavi M, Mirjalili BF, Dehghani Ashkezari M, Dadfar F, Mohaghegh N, Emami S, Salehi F, Nadri H, Ardestani SK, Firoozpour L, Khoobi M, Foroumadi A
Eur. J. Med. Chem, Vol.127, Year. 2017,
48.

Synthesis and biological evaluation of 5-amino-2-phenyl-4H-pyrano[2,3-b]quinoline-3-carboxylates


Authors: Eghtedari M, Sarrafi Y, Nadri H, Mahdavi M, Moradi A, Homayouni Moghadam F, Emami S, Firoozpour L, Asadipour A, Sabzevari O, Foroumadi A
Eur. J. Med. Chem, Vol.128, Year. 2017,
49.

Synthesis and biological evaluation of 1,3,4-thiadiazole linked phthalimide derivatives as anticancer agents


Authors: Rezaeia Z, Moghimi S, Javaheri R, Asadi M, Mahdavi M, Shabani S, Edraki N, Firuzi O, Safavi M, Aminia M, Asadipour A, Zeinalzadeh E, Firoozpour L, Foroumadi A.
letters in drug design and discovery, Vol.14, No.10, Year. 2017,
Download
50.

Protective effects of physical exercise on MDMA-induced cognitive and mitochondrial impairment


Authors: Taghizadeh G, Pourahmad J, Mehdizadeh H, Foroumadi A, Torkaman-Boutorabi A, Hassani S, Naserzadeh P, Shariatmadari R, Gholami M, Rouini MR, Sharifzadeh M
Free Radic. Biol. Med , Vol.99, Year. 2016, Page:11-19,
51.

Design and synthesis of novel anti-Alzheimer’s agents: Acridine-chromenone and quinoline-chromenone hybrids


Authors: Najafi Z, Saeedi M, Mahdavi M, Sabourian R, Khanavi M, Tehrani MB, Moghadam FH, Edraki N, Karimpor-Razkenari E, Sharifzadeh M, Foroumadi A, Shafiee A, Akbarzadeh T.
Bioorg. Chem, Vol.67, Year. 2016, Page:84-94,
52.

Transition-Metal-Catalyzed Acyloxylation: Activation of C(sp2)–H and C(sp3)–H Bonds


Authors: Moghimi S, Mahdavi M, Shafiee A, Foroumadi A
Eur. J. Org. Chem, Vol.20, Year. 2016, Page:3282-3299,
53.

Protective effect of pentoxifylline on male Wistar rat testicular germ cell apoptosis induced by 3,4-methylenedioxymeth amphetamine.


Authors: Nouri M, Movassaghi S, Foroumadi A, Soleimani M, Sharifi ZN
Iran J. Basic Med. Sci, Vol.19, Year. 2016, Page:646-652,
54.

Synthesis and anticholinesterase activity of coumarin-3-carboxamides bearing tryptamine moiety


Authors: Ghanei-Nasab S, Khoobi M, Hadizadeh F, Marjani A, Moradi A, Nadri H, Emami S, Foroumadi A, Shafiee A
Eur. J. Med. Chem, Vol.121, Year. 2016, Page:40-46,
55.

Synthesis and structure-activity relationship study of tacrine-based pyrano[2,3-c]pyrazoles targeting AChE/BuChE and 15-LOX


Authors: Pourabdi L, Khoobi M, Nadri H, Moradi A, Moghadam FH, Emami S, Mojtahedi MM , Haririan I, Forootanfar H, Ameri A, Foroumadi A, Shafiee A.
Eur. J. Med. Chem, Vol.123, Year. 2016, Page:298-308,
56.

CuBr/Et3N-Promoted Reactions of 2-Aminobenzamides and Isothiocyanates: Efficient Synthesis of Novel Quinazolin-4(3H)-ones


Authors: Mahdavi M, Asadi A, Khoshbakht M, Saeedi M, Bayat M, Foroumadi A, Shafiee A.
Helvetica Chimica Acta, Vol.99, Year. 2016, Page:378-383,
57.

An Efficient Four-Step Approach Toward Fused Triazino[1,6-a] Quinazolines


Authors: Sayahi MH , Baghersaei S, Goli F, Moghimi S, Mahdavi M, Firoozpour L, Shafiee A, Foroumadi A
Comb. Chem. High Throughput Screen, Vol.19, Year. 2016, Page:189-192,
58.

QSAR and docking studies on the (5-nitroheteroaryl-1,3,4-thiadiazole-2-yl) piperazinyl analogs with antileishmanial activity


Authors: Tahghighi A, Hamzeh-Mivehroud M, Asadpour Zeynali K, Foroumadi A, Dastmalchi S.
Journal of Chemometrics , Vol.30, Year. 2016, Page:284-293,
59.

Synthesis and cytotoxicity of novel chromenone derivatives bearing 4-nitrophenoxy phenyl acryloyl moiety


Authors: Mahdavi M, Mohammadi-Izad S, Saeedi M, Safavi M, Sadat Ebrahimi SE, Foroumadi A, Shafiee A
Journal of the Iranian Chemical Society, Vol.13, Year. 2016, Page:1139-1144,
60.

Synthesis and evaluation of novel quinazolinone-1,2,3-triazoles as inhibitors of lipoxygenase


Authors: Farjadmand F, Arshadi H, Moghimi S, Nadri H, Moradi A, Eghtedari M, Jafarpour F, Mahdavi M, Shafiee A, Foroumadi A.
Journal of Chemical Research, Vol.40, Year. 2016, Page:188-191,
61.

The importance of triazole scaffold in the development of anticonvulsant agents


Authors: Ayati A, Emami S, Foroumadi A
Eur. J. Med. Chem, Vol.109, Year. 2016, Page:380-392,
62.

A novel and efficient synthesis of 2-substituted quinazolin-4(3H)-ones by the reaction of (het)arylmethanamines with isatoic anhydride


Authors: Mahdavi M, Hassanzadeh R, Soheilizad M, Golshani S, Moghimi S, Firoozpour L, Shafiee A, Foroumadi A.
Tet. Lett , Vol.57, Year. 2016, Page:3770-3772,
63.

Phthalimide-Derived N-Benzylpyridinium Halides Targeting Cholinesterases: Synthesis and Bioactivity of New Potential Anti-Alzheimer's Disease Agents


Authors: Saeedi M, Golipoor M, Mahdavi M, Moradi A, Nadri H, Emami S, Foroumadi A, Shafiee A.
Arch. Pharm. (Weinheim) , Vol.349, Year. 2016, Page:293-301,
64.

An Efficient Three-Step Synthesis of Benzo [e] Imidazo [1, 2-c][1, 2, 3] Triazines.


Authors: Pilali H, Faraji Kamazani Sh, Moradi Sh, Moghimi S, Mahdavi M, Firoozpour L, Shafiee A, Foroumadi A
Synthetic Communications, Vol.46, Year. 2016, Page:563-567,
65.

Synthesis and Cytotoxic Evaluation of Novel1,2,3‐Triazole‐4‐Linked(2E,6E)‐2‐Benzylidene‐6‐(4‐nitrobenzylidene) cyclohexanones


Authors: Mahdavi M, Akhbari M, Saeedi M, Karimi M, Foroughi N, Karimpour‐Razkenari E, Alinezhad H, Foroumadi A, Shafiee A, Akbarzadeh T
Helvetica Chimica Acta , Vol.99, Year. 2016, Page:175-180,
66.

Design, synthesis, and biological evaluation of new series of 2-amido-1,3,4-thiadiazole derivatives as cytotoxic agents.


Authors: Almasirad A, Firoozpour L, Nejati M, Edraki N, Firuzi O, Khoshneviszadeh M, Mahdavi M, Moghimi S, Safavi M, Shafiee A, Foroumadi A.
Zeitschrift für Naturforschung B , Vol.71, Year. 2016, Page:205-210,
67.

In-vitro Antibacterial Evaluation of Some Fluoroquinolone Derivatives Against Food Borne Bacteria


Authors: Shariatifar N, Rezaei M, Sayadi M, Moshafi MH, Saeedi M,. Mohammadhosseini N, Moghimi S, Foroumadi A.
Journal of Sciences, Islamic Republic of Iran, Vol.27, Year. 2016, Page:129-133,
68.

A Novel Copper-Catalyzed preparation of pyrido [1, 2-a] pyrimidine derivatives.


Authors: Mahdavi M, Fazli Estabragh R, Moghimi S, Sayahi MH, Shafiee A, Foroumadi A.
synlett, Vol.27, Year. 2016, Page:1359-1362,
69.

Design, synthesis, pharmacological evaluation, and docking study of new acridone-based 1,2,4-oxadiazoles as potential anticonvulsant agents


Authors: Mohammadi-Khanaposhtani M, Shabani M, Faizi M, Aghaei I, Jahani R, Sharafi Z, Shamsaei Zafarghandi N, Mahdavi M, Akbarzadeh T, Emami S, Shafiee A, Foroumadi A.
Eur. J. Med. Chem, Vol.112, Year. 2016, Page:91-98,
70.

Iodine-Mediated Synthesis of Novel Pyrazole Derivatives


Authors: Mahdavi M, Khoshbakht M, Saeedi M, Asadi M, Bayat M, Foroumadi A, Shafiee A.
Synthesis , Vol.48, Year. 2016, Page:541-546,
71.

Discovery of novel dual inhibitors against Mdm2 and Mdmx proteins by in silico approaches and binding assay


Authors: Golestanian S, Sharifi A, Popowicz GM, Azizian H, Foroumadi A, Szwagierczak A, Holak TA, Amanlou M
Life Sciences, Vol.145, Year. 2016, Page:240-246,
72.

Treatment of Helicobacter pylori infection: Current and future insights


Authors: Safavi M, Sabourian R, Foroumadi A
World Journal of Clinical Cases , Vol.4, Year. 2016, Page:5-19,
73.

Sulfonic Acid Supported Phosphonium Based Ionic Liquid Functionalized SBA-15 for the Synthesis of 2-Amino-3-cyano-4,6-diarylpyridines


Authors: Ma'mani L, Hajihosseini E, Saeedi M, Mahdavi M, Asadipour A, Firoozpour L, Shafiee A , Foroumadi A
Synthesis and Reactivity in Inorganic, Metal Organic and Nano Metal Chemistry , Vol.46, Year. 2016, Page:306-310,
74.

efficacy of Iranian traditional and folk medicinal plants for some gastroduodenal disorders


Authors: Safavi M, shams-Ardakani M.R, seyed bagheri M.S, Foroumadi A
Trenditional and Integrative Medicine , Vol.1, Year. 2016, Page:3-17,
75.

Anticonvulsant activity of 1,2,4-triazine derivatives with pyridyl side chain: synthesis, biological, and computational study.


Authors: Hamid Irannejad, Hamid Nadri, Nima Naderi, Seyedeh Nesa Rezaeian, Neda Zafari, Alireza Foroumadi, Mohsen Amini, Mehdi Khoobi
Med Chem Res, Vol.24, Year. 2015, Page:2505-2513,
76.

Synthesis and In Vitro Cytotoxic Activity of Novel Triazole-Isoxazole Derivatives.


Authors: Zahra Najafi, Mohammad Mahdavi, Maliheh Safavi, Mina Saeedi, Heshmatollah Alinezhad, Mahboobeh Pordeli, Sussan Kabudanian Ardestani, Abbas Shafiee, Alireza Foroumadi, Tahmineh Akbarzadeh
J. Heterocyclic Chem, Vol.52, Year. 2015,
77.

Synthesis of Novel Dibenzylbutyrolactones as Dimethylmatairesinol Analogues


Authors: Babak Heidary Alizadeh, Alireza Foroumadi, Farzad Kobarfard, Mina Saeedi, Abbas Shafiee.
J. Heterocyclic Chem, Vol.52, Year. 2015,
78.

Synthesis of Novel 2-Oxoquinoline Derivatives via Ugi-Four-Component-Heck Reaction


Authors: Mohammad Ali Rasouli, Mohammad Mahdavi, Mina Saeedi, Parviz Rashidi Ranjbar, Abbas Shafiee, Alireza Foroumadi
J. Heterocyclic Chem, Vol.52, Year. 2015,
79.

Efficient Synthesis of Novel Thiazol-2-ylidene-amides Using Carbonylthiourea Building Blocks


Authors: Mina Saeedi, Fereshteh Goli, Mohammad Mahdavi, Ali Asadipour, Abbas Shafiee, Alireza Foroumadi
J. Heterocyclic Chem, Vol.52, Year. 2015,
80.

-Synthesis and Evaluation of Ethyl 2,4-dioxo-4- arylbutanoate Derivatives as Src Kinase Inhibitors.


Authors: A. Rafinejad, A. Fallah-Tafti, R. Tiwari, A. Nasrolahi Shirazi D. Mandal, K. Parang, A. Foroumadi, T. Akbarzadeh
Journal of Sciences, Islamic Republic of Iran, Vol.26, Year. 2015,
81.

Brønsted Acidic Phosphonium Based Ionic Liquid Functionalized SBA-15 [HO3S-PhospIL@SBA-15]: Green, Recyclable, and Efficient Catalyst for the Synthesis of Pyrano[3,2-c]Chromenone Derivatives.


Authors: Mina Saeedi, Mohammad Jeiroudi, Leila Mamani, Mohammad Mahdavi, Eskandar Alipour, Abbas Shafiee, Alireza Foroumadi
Iran.J.Chem.Chem. Eng , Vol.34, Year. 2015,
82.

Design , synthesis, biological evaluation and docking studyof acetylcholinesterase inhibitors : new acridone -1,2,4-oxadiazole-1,2,3-triazole hybrids.


Authors: Maryam Mohammadi-Khanaposhtani, Mohammad Mahdavi, Mina Saeedi, Reyhaneh Sabouriyan, Maliheh Safavi, Mahnaz Khanavi, Alireza Foroumadi, Abbas Shafiee, Tahmineh Akbarzadeh
Chemical biology and drug design , Vol.86, Year. 2015,
83.

Design, Synthesis, in vitro cytotoxic activity evaluation and apoptosis -induction study of new 9(10H)-acridinone -1,2,3-triazoles.


Authors: Maryam Mohammadi khanaposhtani , Maliheh Safavi, Reyhaneh Sabouriyan, Mohammad Mahdavi, Mahboobeh Pordeli, Mina Saeedi, Sussan Kaboudanian Ardestani, Alireza Fouromadi, Abbas Shafiee, Tahmineh Akbarzadeh
Molecular Diversity , Vol.19, Year. 2015,
84.

Synthesis of novel 1,2,3-triazol-dihydro[3,2-c] chromenone as acetyl cholinesterase inhibitors.


Authors: Mina Saeedi, Shirin Ansari, Mohammad Mahdavi, Reyhaneh Sabouriyan, Tahmineh Akbarzadeh , Alireza Foroumadi, Abbas Shafiee
Synthetic Communication , Vol.45, Year. 2015,
85.

highly efficient method for the synthesis of novel 1H-spiro[ indone -2,2-quinazoline] -1,3,4(3H) trone derivatives


Authors: Seyed esmail sadat ebrahimi, Soroor Irannezhad, Setareh Moghimi, Azadeh Yahya Meymandi, Mohammad Mahdavi, Abbas shafiee, Alireza Foroumadi
Journal of Chemical Research , Vol.39, Year. 2015,
86.

Cytotoxicity and apoptosis inducing activities of 2-amino 4H- chromene-3- carbonitrile derivatives loaded on gold nanoparticles against human breast cancer cell line T47D


Authors: Zahra Saffari, Maryam Farahnak Zarabi, Hassan Aryapour, Alireza Foroumadi, Ali Farhangi, Soheil Ghassemi, Azim Akbarzadeh
Indian Journal of Clinical Biochemistry,, Vol.30, Year. 2015,
87.

Sulfamic acid -functionalized hydroxyl apatite –encapsulated Y-Fe2O3- nanoparticles as a magnetically recoverable catalyst for synthesis of N-fused imidazole-quinoline conjugates under solvent – free condition


Authors: Arash Mouradzadegun, Leila Mamani, Mohammad Mahdavi, Zahra Rashid , Abbas Shafiee, Alireza Foroumadi, Shima dianat
RSC Advances, Vol.101, Year. 2015,
88.

Cytotoxic activity of some 1-(2,4-dihydroxyphenyl)-3-(4-phenyl piperidin-1-yl)prop-2-en-1-one derivatives using MTT assay.


Authors: Farzaneh Fesahat, Mehdi Khoshneviszadeh , Alireza Foroumadi, Alireza Vahidi, Maryam Fereidounpour, Amirhossin Sakhteman
Trends in Pharmaceutical Sciences, Vol.1, Year. 2015,
89.

Efficient synthesis of 2-methylenethiazolo[ 2,3-b] quinazolinone derivatives.


Authors: Mohammad Mahdavi, Maryam Bialam , Mina Saeedi, Farnaz Jafarpour, Alireza Foroumadi
synlett, Vol.26, Year. 2015,
90.

Synthesis of new benzo [f] imidazo [1, 2-d][1, 4] oxazepines: AgNO 3-mediated intramolecular hydroamination.


Authors: Mohammad Mahdavi, Roshanak Hariri, Mina Saeedi, Alireza Foroumadi, Abbas Shafiee, Tahmineh Akbarzadeh
Tetrahedron letters,, Vol.59, Year. 2015,
91.

Synthesis and evaluation of novel oxoisoindoline derivatives as acetylcholinesterase inhibitors.


Authors: Ayeh Rayatzadeh, Mina Saeedi, Mohammad Mahdavi, Zahra Rezaei, Reyhaneh Sabourian, Mohammad Hossein Mosslemin, Tahmineh Akbarzadeh, Alireza Foroumadi,Abbas Shafiee
Monatshefte für Chemie, Vol.146, Year. 2015,
92.

Combined isocyanide-based multi-component Ullmann-type reaction: an efficient access to novel nitrogen-containing pentacyclic compounds


Authors: Shima Dianat, Mohammad Mahdavi, Setareh Moghimi, Arash Mouradzadegun, Abbas Shafiee, Alireza Foroumadi
Molecular Diversity, Vol.19, Year. 2015,
93.

Synthesis and structure-activity relationship study of benzofuranbased chalconoids bearing benzylpyridinium moiety as potent acetylcholinesterase inhibitors


Authors: Manizheh Mostofi, Ghodsi Mohammadi Ziarani, Mohammad Mahdavi, Alireza Moradi, Hamid Nadri, Saeed Emami, Heshmatollah Alinezhad, Alireza Foroumadi, Abbas Shafiee
European Journal of Medicinal Chemistry, Vol.103, Year. 2015,
94.

Polyethyleneimine-modified superparamagnetic Fe3O4 nanoparticles: An efficient, reusable and water to lerance nanocatalyst.


Authors: Mehdi Khoobi, Tayebeh Modiri Delshad, MohsenVosooghi, Masoumeh Alipour, Hosein Hamadi, Eskandar Alipour, Morteza PiraliHamedani, Seyed Esmaeil Sadatebrahimi, Zahra Safaei, Alireza Foroumadi, Abbas Shafiee
Journal of Magnetism and Magnetic Materials, Vol.375, Year. 2015,
95.

Synthesis of some novel pyrano [2,3-f] chromenone derivatives


Authors: Babak Heidary Alizadeh, Mina Saeedi, Gholamreza Dehghan, Alireza Foroumadi, Abbas Shafiee.
Journal of the Iranian Chemical Society, Vol.12, Year. 2015,
96.

A structural model of the anaphase promoting complex co-activator (Cdh1) and insilico design of inhibitory compounds.


Authors: H. Rahimi, B. Negahdari, M.A. Shokrgozar, A. Madadkar-Sobhani, R. Mahdian1, A. Foroumadi, M. Kafshdouzi Amin and M. Karimipoor
Research in Pharmaceutical Sciences, Vol.10, Year. 2015,
97.

Synthesis and biological evaluation of 5-benzylidenerhodanine-3-acetic acid derivatives as AChE and 15-LOX inhibitors


Authors: Negah Shafii, Mehdi Khoobi, Mohsen Amini, Amirhossein Sakhteman, Hamid Nadri, Alireza Moradi, Saeed Emami, Ebrahim Saeedian Moghadamb, Alireza Foroumadi , Abbas Shafiee.
Journal of Enzyme Inhibition and Medicinal Chemistry,, Vol.30, No.3, Year. 2015,
98.

Synthesis and Evaluation of Chroman-4-One Linked to N-Benzyl Pyridinium Derivatives as New Acetylcholinesterase Inhibitors


Authors: Saman Arab, Seyed-Esmail Sadat-Ebrahimi, Maryam Mohammadi-Khanaposhtani, Alireza Moradi, Hamid Nadri, Mohammad Mahdavi, Setareh Moghimi, Mehdi Asadi, Loghman Firoozpour, Morteza Pirali-Hamedani, Abbas Shafiee and Alireza Foroumadi
Archive der pharmazie, Vol.348, No.9, Year. 2015,
99.

minimal structural requirements, molecular dynamics simulations, and the effect of piperitone on the emergence of nitrofurantoin resistance in Enterobacteriaceae


Authors: Shahverdi AR, Mirzaie S, Rafii F, Kakavand M, Foroumadi A
Journal of molecular modeling, Vol.21, No.198, Year. 2015,
100.

Efficient multi-component synthesis of 1,4-benzodiazepine-3,5-diones: a Petasis-based approach


Authors: Saeedeh Noushini, Mohammad Mahdavi, Loghman Firoozpour, Setareh Moghimi, Abbas Shafiee, Alireza Foroumadi
Tetrahedron,, Vol.71, No.36, Year. 2015,
101.

Straightforward Approach Toward Dihydrothiazoles via Intramolecular Bromocyclization.


Authors: Seyed Esmail Sadat-Ebrahimi, Marzieh Ganjizadeh Zarj, Setareh Moghimi, Azadeh Yahya-Meymandi, Mohammad Mahdavi, Saman Arab, Abbas Shafiee and Alireza Foroumad
Synthetic Communication, Vol.45, No.18, Year. 2015,
102.

Novel 1,2,3,4-Tetrahydroquinazolinones via Reaction of 2-Amino-N-substituted Benzamides and Dimethyl Acetylenedicarboxylate


Authors: Semiramis Nahavandian, Sadegh Allameh, Mina Saeedi, Shirin Ansari, Mohammad Mahdavi, Alireza Foroumadi and Abbas Shafiee
Helvetica Chimica Acta, Vol.98, No.7, Year. 2015,
103.

Medicinal plants in the treatment of Helicobacter pylori infections


Authors: Maliheh Safavi, Mohammadreza Shams Ardakani, Alireza Foroumadi
Pharm Biol, Vol.53, No.7, Year. 2015,
104.

Design, synthesis and anticholinesterase activity of novel benzylidenechroman-4-ones bearing cyclic amine side chain


Authors: Yaghoub Pourshojaei, Ali Gouranourimi , Shohre Hekmat, Ali Asadipour, Samira Rahmani-Nezhad, Alireza Moradi, Hamid Nadri, Farshad Homayouni Moghadam, Saeed Emami, Alireza Foroumadi, Abbas Shafiee
European Journal of Medicinal Chemistry, Vol.97, Year. 2015,
105.

New tetracyclic tacrine analogs containing pyrano[2,3-c]pyrazole: Efficient synthesis, biological assessment and docking simulation Study.


Authors: Mehdi Khoobi, Farzaneh Ghanoni, Hamid Nadri, Alireza Moradi, Morteza Pirali Hamedani, Farshad Homayouni Moghadam, Saeed Emami, Mohsen Vosooghi, Reza Zadmard, Alireza Foroumadi, Abbas Shafiee.
European Journal of Medicinal Chemistry , Vol.89, Year. 2015,
106.

Novel N-2-(Furyl)-2-(chlorobenzyloxyimino) ethyl Piperazinyl Quinolones: Synthesis, Cytotoxic Evaluation and Structure-activity Relationship


Authors: Negar Mohammadhosseini, Mahboobeh Pordeli, Maliheh Safavi, Loghman Firoozpour, Fatame Amin, Sussan Kabudanian Ardestani, Najmeh Edrakif, Abbas Shafiee and Alireza Foroumadi
Iranian Journal of Pharmaceutical Research, Vol.14, No.4, Year. 2015,
107.

Synthesis and anticancer activity of N-substituted 2-arylquinazolinones bearing trans-stilbene scaffold


Authors: Mohammad Mahdavi, Keyvan Pedrood, Maliheh Safavi, Mina Saeedi, Mahboobeh Pordeli, Sussan Kabudanian Ardestani, Saeed Emami, Mehdi Adib, Alireza Foroumadi, Abbas Shafiee
European Journal of Medicinal Chemistry,, Vol.95, Year. 2015,
108.

Synthesis and anticholinergic activity of 4‐hydroxycoumarin derivatives containing substituted benzyl‐1, 2, 3‐triazole moiety.


Authors: Sahar Mohammad Bagheri, Mehdi Khoobi, Hamid Nadri, Alireza Moradi, Saeed Emami, Leili Jalili‐Baleh, Farnaz Jafarpour, Farshad Homayouni Moghadam, Alireza Foroumadi, Abbas Shafiee
Chemical Biology & Drug Design., Year. 2015,
109.

9H‐Carbazole Derivatives Containing the N‐Benzyl‐1, 2, 3‐triazole Moiety as New Acetylcholinesterase Inhibitors.


Authors: Hamidreza Akrami, Bibi F Mirjalili, Mehdi Khoobi, Alireza Moradi, Hamid Nadri, Saeed Emami, Alireza Foroumadi, Mohsen Vosooghi, Abbas Shafiee
Archiv der Pharmazie, Vol.348, No.5, Year. 2015,
110.

N‐(2‐(Piperazin‐1‐yl) phenyl) arylamide Derivatives as β‐Secretase (BACE1) Inhibitors: Simple Synthesis by Ugi Four‐Component Reaction and Biological Evaluation.


Authors: Najmeh Edraki, Omidreza Firuzi, Yousef Fatahi, Mohammad Mahdavi, Mehdi Asadi, Saeed Emami, Kouros Divsalar, Ramin Miri, Aida Iraji, Mehdi Khoshneviszadeh, Loghman Firoozpour, Abbas Shafiee, Alireza Foroumadi
Archive der pharmazie, Vol.348, No.5, Year. 2015,
111.

.Recent applications of 1, 3-thiazole core structure in the identification of new lead compounds and drug discovery


Authors: Adile Ayati, Saeed Emami, Ali Asadipour, Abbas Shafiee, Alireza Foroumadi
European journal of medicinal chemistry, Vol.97, Year. 2015,
112.

Synthesis of novel 5-arylidene (thio) barbituric acid and evaluation of their urease inhibitory activity.


Authors: Mohsen Vosooghi , Soghra Farzipour , Mina Saeedi , Neda Babazadeh Shareh , Mohammad Mahdavi , Shabnam Mahernia , Alireza Foroumadi , Massoud Amanlou , Abbas Shafiee.
Journal of the Iranian Chemical Society , Vol.12, No....., Year. 2015,
113.

Synthesis and cytotoxic activity of novel poly-substituted imidazo [2, 1-c][1, 2, 4] triazin-6-amines


Authors: Tahmineh Akbarzadeh, Saeedeh Noushini, Somayeh Taban, Mohammad Mahdavi, Mahsima Khoshneviszadeh, Mina Saeedi, Saeed Emami, Mohammad Eghtedari, Yaghoub Sarrafi, Mehdi Khoshneviszadeh, Maliheh Safavi, Kouros Divsalar, Mohammad Hassan Moshafi, Ali Asadipour, Reyhaneh Sabourian, Najmeh Edraki, Omidreza Firouzi, Ramin Miri, Abbas Shafiee, Alireza Foroumadi.
Molecular Diversity, Vol.19, No....., Year. 2015,
114.

Benzofuran-derived benzylpyridinium bromides as potent acetylcholinesterase inhibitors


Authors: Farzaneh Baharloo a, Mohammad Hossein Moslemin a, Hamid Nadri b, Ali Asadipour c, Mohammad Mahdavi d, Saeed Emami e, Loghman Firoozpour f, Razieh Mohebat a, Abbas Shafiee d, Alireza Foroumadi
European Journal Of Medicinal Chemistry, Vol.93, Year. 2015,
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115.

Potent acetylcholinesterase inhibitors: Design, synthesis, biological evaluation, and docking study of acridone linked to 1,2,3-triazole derivatives


Authors: Maryam Mohammadi-Khanaposhtani a, Mina Saeedi b, Narges Shamsaei Zafarghandi a, Mohammad Mahdavi c, Reyhaneh Sabourian d, Elahe Karimpour Razkenari d, Heshmatollah Alinezhad e, Mahnaz Khanavi f, Alireza Foroumadi c, Abbas Shafiee c, Tahmineh Akbarzadeh
European Jornal Of Medicinal Chemistry, Vol.92, Year. 2015,
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116.

SYNTHESIS AND EVALUATION OF COUMARIN– RESVERATROL HYBRIDS AS 15-LIPOXYGENAZE INHIBITORS


Authors: Samira Rahmani-Nezhad,1 Leila Khosravani,1 Mina Saeedi,2 Kouros Divsalar,3 Loghman Firoozpour,4 Yaghoub Pourshojaei,1 Yaghoub Sarrafi,5 Hamid Nadri,6 Alireza Moradi,6 Mohammad Mahdavi,1 Abbas Shafiee,1 and Alireza Foroumadi3,4
Syntheytic Communication, Vol.45, Year. 2015,
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117.

Synthesis, antileishmanial activity and QSAR study of (1,3,4- thiadiazol-2-ylthio) acetamides derived from 5-nitrofuran


Authors: Mohsen Vosooghi • Reyhaneh Sabourian • Azar Tahghighi • Mohammad Mahdavi • Saeed Emami • Sepideh Razmi • Sussan Kabudanian Ardestani • Maliheh Safavi • Parham Foroumadi • Sara Kaveh • Mehdi Khoshneviszadeh • Najmeh Edraki • Abbas Shafiee • Alireza Foroumadi
MEDICINAL CHEMISTRY RESEARCH, Vol.24, Year. 2015,
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118.

Simple and efficient syntheses of novel benzo[4,5]imidazo [1,2-a]pyridine derivatives


Authors: Fereshteh Goli-Garmroodi a, Marzieh Omidi b, Mina Saeedi c, Farhad Sarrafzadeh d, Ali Rafinejad c, Mohammad Mahdavi a, Ghasem Rezanejade Bardajee b, Tahmineh Akbarzadeh a,c, Loghman Firoozpour e, Abbas Shafiee a, Alireza Foroumadi a,d,⇑
Tetrahedron letters, Vol.46, Year. 2015,
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119.

Synthesis and Cytotoxic Activity of Some Novel Dihyrobenzo[h]pyrano [3,2-c]chromene Derivatives


Authors: Nasim Esmati,a Mahsa Foroughian,a Mina Saeedi,b Mohammad Mahdavi,b Mehdi Khoshneviszadeh,b,c Omidreza Firuzi,c Nader Tanideh,c Ramin Miri,c Najmeh Edraki,b,c Abbas Shafiee,b and Alireza Foroumadia,b*
journal of Heterocyclic Chenmistry, Vol.52, Year. 2015,
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120.

Design, synthesis, docking study and cytotoxic activity evaluation of some novel letrozole analogs


Authors: Mohsen Vosooghi1, Loghman Firoozpour2, Abolfazl Rodaki2, Mahboobeh Pordeli3, Maliheh Safavi4,
DARU Journal of pharmaceutical sciences, Vol.22, No.83, Year. 2014,
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121.

Imidazo[2,1-b]thiazole derivatives as new inhibitors of 1,5- lipoxygenase


Authors: Maliheh Barazandeh Tehrani, Saeed Emami, Mehdi Asadi, Mina Saeedi,
European Journal of Medicinal Chemistry, Vol.87, Year. 2014,
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122.

N-Substituted indole carbohydrazide derivatives: synthesis and evaluation of their antiplatelet aggregation activity.


Authors: Seyedeh Sara Mirfazli, Farzad Kobarfard, Loghman Firoozpour, Ali Asadipour, Marjan Esfahanizadeh, Kimia Tabib, Abbas Shafiee and Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences, Vol.22, No.66, Year. 2014,
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123.

Synthesis, in vitro cytotoxicity and apoptosis inducing study of 2-aryl- 3-nitro-2H-chromene derivatives as potent anti-breast cancer agents


Authors: Samira Rahmani-Nezhad a, Maliheh Safavi b, Mahboobeh Pordeli c, Sussan Kabudanian Ardestani c, Leila Khosravani a, Yaghoub Pourshojaei a, Mohammad Mahdavi a, Saeed Emami d, Alireza Foroumadi a, Abbas Shafiee
European Journal of Medicinal Chemistry, Vol.86, Year. 2014, Page:562e569,
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124.

Mixed micellar nanoparticles based on PCL-PEG-PPO-PEG-PCL pentablocks


Authors: Salman Hassanzadeh & Sepideh Khoee & Vahid Farrokhi & Mohamad Mahdavi & Alireza Foroumadi
J Polym Res, Vol.21, Year. 2014, Page:508,
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125.

Synthesis and Anti-Cancer Activity Evaluation of New Dimethoxylated Chalcone and Flavanone Analogs


Authors: Shima H. M. E. Ketabforoosh1, Asma Kheirollahi2, Maliheh Safavi3, Nasim Esmati4, Sussan K. Ardestani2, Saeed Emami5, Loghman Firoozpour4, Abbas Shafiee6, and Alireza Foroumadi4,6
Archive der Pharmazie, Vol.2014, 347, 1–8, Year. 2014,
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126.

Cytotoxicity of some 1-(2,4-dihydroxyphenyl)-3-(4-phenylpiperidin-1-yl) prop-2-en-1-one derivatives using MTT assay


Authors: , Farzaneh Fesahat1, Mehdi Khoshneviszadeh2, Alireza Foroumadi3, AlirezaVahidi1, Maryam Fereidounpour1, Amirhossein Sakhteman2*
Trends in Pharmaceutical Sciences, Vol.2014; 1(1): 15-19; art. 1, No.1, Year. 2014,
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127.

Synthesis of novel 5-phenylimidazo[1,2-c]quinazolin-3-amine derivatives via Groebke–Blackburn–Bienayme multicomponent reaction


Authors: Tahmineh Akbarzadeh, Mohammad Mahdavi, Abolfath Ebrahimi, Alireza Foroumadi, Mina Saeedi, Abbas Shafiee
Monatsh Chem, Vol.145, Year. 2014,
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128.

N-Phenyl-2-p-tolylthiazole-4-carboxamide derivatives: Synthesis and cytotoxicity evaluation as anticancer agents.


Authors: Ahmad Mohammadi-Farani, Alireza Foroumadi, Monireh Rezvani Kashani, Alireza Aliabadi.
Iranian Journal of Basic Medical Sciences , Vol.17, No.7, Year. 2014,
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129.

Synthesis of Novel Benzo[6,7][1,4]oxazepino[4,5-a]quinazolinone Derivatives via Transition-Metal-Free Intramolecular Hydroamination.


Authors: Mohammad Mahdavi, Niloufar Foroughi, Mina Saeedi, Maryam Karimi, Heshmatollah Alinezhad, Alireza Foroumadi, Abbas Shafiee, Tahmineh Akbarzadeh
SYNLETT, Vol.25, Year. 2014, Page:0385–0388,
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130.

Curcumin-loaded guanidine functionalized PEGylated I3ad mesoporous silica nanoparticles KIT-6: Practical strategy for the breast cancer therapy.


Authors: Leila Ma'mani, Safoora Nikzad, Hamidreza Kheiri-manjili, Sharafaldin al-Musawi, Mina Saeedi, Sonia Askarlou, Alireza Foroumadi, Abbas Shafiee.
European Journal of Medicinal Chemistry, Vol.83, Year. 2014,
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131.

Indolinone-based acetylcholinesterase inhibitors: Synthesis, biological activity and molecular modeling.


Authors: Hamidreza Akrami, Bibi Fatemeh Mirjalili, Mehdi Khoobi, Hamid Nadri, Alireza Moradi, Amirhossein Sakhteman, Saeed Emami, Alireza Foroumadi, Abbas Shaee.
European Journal of Medicinal Chemistry, Vol.84, Year. 2014, Page:375-381,
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132.

In vitro antitumor evaluation of 4H-chromene-3-carbonitrile derivatives as a new series of apoptotic inducers.


Authors: Zahra Saffari, Hassan Aryapour , Azim Akbarzadeh, Alireza Foroumadi, Najmeh Jafari, Maryam Farahnak Zarabi, Ali Farhangi
Tumor Biol, Vol.35, Year. 2014, Number of Page:5845–5855
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133.

fficient Solvent-Free Synthesis of Benzothiazine-Fused Pyrrolo[3,4-c]coumarins: Cycloaddition Reactions between Coumarin-Based Dihydro benzothiazoles and Isocyanides.


Authors: Mehdi Khoobi, Ali Ramazani, Mohammad Mahdavi, Alireza Foroumadi, Saeed Emami, Sang Woo Joo, Katarzyna S´ lepokuraf, Tadeusz Lisf, and Abbas Shafiee.
Helvetica Chimica Acta., Vol.97, Year. 2014, Number of Page:847- 853
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134.

Synthesis, biological evaluation and docking study of 3-aroyl-1-(4-sulfamoylphenyl) thiourea derivatives as 15-lipoxygenase inhibitors.


Authors: Mohammad Mahdavi, Maryam Shahzad Shirazi, Raana Taherkhani, Mina Saeedi, Eskandar Alipour, Farshad Homayouni Moghadam, Alireza Moradi, Hamid Nadri, Saeed Emami, Loghman Firoozpour, Abbas Shafiee, Alireza Foroumadi
European Journal of Medicinal Chemistry, Vol.82, Year. 2014,
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135.

Synthesis and cytotoxic evaluation of some new [1,3]dioxolo[4,5-g]chromen-8-one derivatives


Authors: Eskandar Alipour, Zinatsadat Mousavi, Zahra Safaei, Mahboobeh Pordeli, Maliheh Safavi, Loghman Firoozpour, Negar Mohammadhosseini, Mina Saeedi, Sussan Kabudanian Ardestani, Abbas Shafiee and Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences 2014, 22:41, Vol.22, No.41, Year. 2014,
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136.

Synthesis and psychobiological evaluation of modafinil analogs in mice.


Authors: Arezou Lari, Isaac Karimi, Hadi Adibi, Alireza Aliabadi, Loghman Firoozpour and Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences , Vol.21, Year. 2014,
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137.

Antinociceptive properties of new coumarin derivatives bearing substituted 3, 4-dihydro-2Hbenzothiazines.


Authors: Masoumeh Alipour, Mehdi Khoobi, Saeed Emami, Saeed Fallah-Benakohal, Seyedeh Farnaz Ghasemi-Niri, Mohammad Abdollahi, Alireza Foroumadi and Abbas Shafiee.
DARU Journal of Pharmaceutical Sciences, Year. 2014,
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138.

Palladium-catalyzed oxidative CeH bond coupling of indoles


Authors: Ebrahim Kianmehr a,*, Shahrzad Kazemi a, Alireza Foroumadi
Tetrahedron, Vol.70, Year. 2014,
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139.

Imidazolylchromanones containing alkyl side chain as lanosterol


Authors: Saeed Emami, Touba Banipoulad, Hamid Irannejad, Alireza Foroumadi, Mehraban Falahati, Mahtab Ashrafi-Khozani, and Somaye Sharifynia
J Enzyme Inhib Med Chem, Vol. 29(2), Year. 2014, Page:263–271,
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140.

One-pot, four-component synthesis of novel cytotoxic agents 1-(5-aryl-1,3,4-oxadiazol-2-yl)-1-(1H-pyrrol-2-yl)methanamines


Authors: Ali Ramazani, Mehdi Khoobi, Azar Torkaman, Fatemeh Zeinali Nasrabadi, Hamid Forootanfar, Mojtaba Shakibaie, Mandana Jafari, Alieh Ameri, Saeed Emami, Mohammad Ali Faramarzi, Alireza Foroumadi, Abbas Shafiee
European Journal of Medicinal Chemistry , Vol.78, Year. 2014, Number of Page:151-156
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141.

An efficient synthesis of novel dihydrothiazol-2-yl-amides via cyclisation of propargylic carbamothioyl-amides


Authors: Mina Saeedi, Fereshteh Goli, Mohammad Mahdavi, Pouria Sarihi, Ali Asadipour, Abbas Shafieea and Alireza Foroumadi
Journal Of Chemical Research , Vol.38, Year. 2014, Page:131–133,
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142.

Antinociceptive properties of new coumarin derivatives bearing substituted 3,4-dihydro-2Hbenzothiazines


Authors: Masoumeh Alipour, Mehdi Khoobi, Saeed Emami, Saeed Fallah-Benakohal, Seyedeh Farnaz Ghasemi-Niri, Mohammad Abdollahi, Alireza Foroumadi and Abbas Shafiee
DARU Journal of Pharmaceutical Sciences 2014, Vol.22, Year. 2014,
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143.

Convenient and sequential one-pot route for synthesis of 2-thioxoquinazolinone and quinazolinobenzothiazinedione derivatives


Authors: Mehdi Asadi, Shiva Masoomi, Seyed Mostafa Ebrahimi, Mohammad Mahdavi, Mina Saeedi, Abbas Shafiee, Alireza Foroumadi
Monatshefte für Chemie - Chemical Monthly, Vol.145, Year. 2014, Page:497–504,
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144.

Microwave-assisted synthesis and anticonvulsant activity of 5,6-bisaryl-1,2,4-triazine-3-thiol derivatives.


Authors: Hamid Irannejad, Nima Naderi, Saeed Emami, Roja Qobadi Ghadikolaei, Alireza Foroumadi, Tina Zafari, Ali Mazar-Atabaki, Sakineh Dadashpour.
Medicinal Chemistry Research, Vol.23 , Year. 2014, Page:2503–2514,
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145.

Vilsmeler Reagent: An Efficient Reagent For The Transformation Of 2-Aminobenzamides into Quinozoline-4(3H)-One Derivatives.


Authors: Soghra Farzipour, Mina Saeedi, Mohammad Mahdavi, Hossein Yavari, Mohammadreza Mirzahekmati, Nasser Ghaemi, Alireza Foroumadi and Abbas Shafiee
Synthetic Communications, Vol.44, Year. 2014, Page:481–487,
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146.

Synthesis and evaluation of antiproliferative activity of substituted N-(9-oxo-9H-xanthen-4-yl)benzenesulfonamides.


Authors: Somayeh Motavallizadeh, Asal Fallah-Tafti, Saeedeh Maleki, Amir Nasrolahi Shirazi, Mahboobeh Pordeli, Maliheh Safavi, Sussan Kabudanian Ardestani, Shaaban Asd, Rakesh Tiwari, Donghoon Oh, Abbas Shafiee, Alireza Foroumadi, Keykavous Parang, Tahmineh Akbarzadeh
Tetrahedron Letters, Vol.373–375 , Year. 2014, Page:373–375 ,
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147.

Green and Catalyst-free One-pot Synthesis of Anthraniamide Schiff Base: an Approch Toward Sirttinol


Authors: Seyed Mostafa Ebrahimi, Mohammad Mahdavi, Saeed Emami, Mina Saeedi, Mehdi Asadi, Loghman Firoozpour, Mehdi Khoobi, Kouros Divsalar,Abbas Shafiee, and Alireza Foroumadi.
Synthetic Communications, Vol. 244, Year. 2014, Page:665–673,
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148.

Synthesis and In vitro cytotoxic activity evaluation of (E)-16-(substituted benzylidene) derivatives of dehydroepiandrosterone.


Authors: Mohsen Vosooghi, Hoda Yahyavi1, Kouros Divsalar, Hashem Shamsa1, Asma Kheirollahi, Maliheh Safavi, Sussan Kabudanian Ardestani, Sareh Sadeghi-Neshat, Negar Mohammadhosseini, Najmeh Edraki, Mehdi Khoshneviszadeh, Abbas Shafiee and Alireza Foroumadi.
DARU Journal of Pharmaceutical Sciences, Vol.21(34), Year. 2013,
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149.

Activity of 2-(2-(4-(2-Oxo-2-phenylethyl)piperazin-1-yl) ethyl)Isoindoline-1,3-dione Derivatives with Potential Anti-Alzheimer Effects.


Authors: Alireza Aliabadi, Alireza Foroumadi, Ahmad Mohammadi-Farani, Mahdi Garmsiri Mahvar
Iranian Journal of Basic Medical Sciences, Vol.16(10), Year. 2013, Page:1049- 1054,
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150.

The importance of synthetic drugs for type 2 diabetes drug discovery.


Authors: Maliheh Safavi, Alireza Foroumadi & Mohammad Abdollahi
Expert Opin. Drug Discov, Vol.8, No.11, Year. 2013, Number of Page:1339-1363
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151.

Synthesis and psychobiological evaluation of modafinil analogs in mice.


Authors: Arezou Lari, Isaac Karimi, Hadi Adibi, Alireza Aliabadi, Loghman Firoozpour, and Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences, Vol.21, No.67, Year. 2013,
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152.

Determination of MDMA and Its Three Metabolites in the Rat Perfused Liver.


Authors: Bardia Jamali, Yalda Hosseinzadeh Ardakani, Alireza Foroumadi, Farzad Kobarfard, Mohammad-Reza Rouini
Journal of Analytical Toxicology, Vol.37, No.6, Year. 2013, Number of Page:357-61
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153.

Synthesis of novel fused 4,5-dihydro-1,2,3-triazolo[1,5-a][1,4] benzodiazepine derivatives via four-component UgieSmiles-type reaction.


Authors: Mina Saeedi, Mohammad Mahdavi, Alireza Foroumadi, Abbas Shafiee.
Tetrahedron, Vol.69, Year. 2013, Number of Page:3506-3510
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154.

Synthesis and evaluation of 4-substituted coumarins as novel acetylcholinesterase inhibitors


Authors: Seyyede Faeze Razavi, Mehdi Khoobi, Hamid Nadri, Amirhossein Sakhteman, Alireza Moradi, Saeed Emami, Alireza Foroumadi, Abbas Shafiee
European Journal of Medicinal Chemistry, Vol.64, Year. 2013, Number of Page:252-259
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155.

2-Amino-4-(nitroalkyl)-4H-chromene-3-carbonitriles as New Cytotoxic Agents.


Authors: Afsaneh Zonouzi, Roghieh Mirzazadeh, Maliheh Safavi, Sussan Kabudanian Ardestani, Saeed Emamid and Alireza Foroumadi
Iranian Journal of Pharmaceutical Research, Vol.12, No.4, Year. 2013, Page:679-685,
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156.

Synthesis and Antidiabetic Evaluation of Benzenesulfonamide Derivatives.


Authors: Nouraddin Hosseinzadeh, Soodeh Seraj, Mohamad Ebrahim Bakhshi-Dezffoli, Mohammad Hasani, Mehdi Khoshneviszadeh, Saeed Fallah-Bonekohal, Mohammad Abdollahi, Alireza Foroumadie and Abbas Shafiee
Iranian Journal of Pharmaceutical Research, Vol.12, Year. 2013, Number of Page:325-330
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157.

Design, synthesis, docking study and biological evaluation of some novel tetrahydrochromeno [3’,4’:5,6] pyrano[2,3-b]quinolin-6(7H)-one derivatives against acetyl- and butyrylcholinesterase


Authors: Mehdi Khoobi, Masoumeh Alipour, Alireza Moradi, Amirhossein Sakhteman, Hamid Nadri, Seyyede Faeze Razavi, Mehdi Ghandi, Alireza Foroumadi, Abbas Shafiee
European Journal of Medicinal Chemistry, Vol.68, Year. 2013, Page:291–300,
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158.

Design, synthesis and biological evaluation of novel anti-cytokine 1,2,4-triazine derivatives.


Authors: Mehdi Khoshneviszadeh, Mohammad H. Ghahremani, Alireza Foroumadi, Ramin Miri, Omidreza Firuzi, Armin Madadkar-Sobhani, Najmeh Edraki, Maliheh Parsa, Abbas Shafiee.
Bioorganic & Medicinal Chemistry, Vol.21, Year. 2013, Page:6708–6717,
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159.

Phenylimino-2H-chromen-3-carboxamide derivatives as novel small molecule inhibitors of b-secretase.


Authors: Najmeh Edraki, Omidreza Firuzi, Alireza Foroumadi, Ramin Miri, Armin Madadkar-Sobhani, Mehdi Khoshneviszadeh, Abbas Shafiee
Bioorganic & Medicinal Chemistry, Vol.21, Year. 2013, Page:2396–2412,
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160.

Synthesis of Some New 3-Coumaranone and Coumarin Derivatives as Dual Inhibitors of Acetyland Butyrylcholinesterase


Authors: Masomeh Alipour, Mehdi Khoobi, Hamid Nadri, Amirhossein Sakhteman, Alireza Moradi, Mehdi Ghandi, Aliraza Foroumadi, Abass Shafiee
Archiv der Pharmazie, Vol.346, Year. 2013, Page:1-11,
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161.

Synthesis and In Vitro Cytotoxic Activity of Novel Chalcone-Like Agents


Authors: Bahram Letafat , Raheleh Shakeri, Saeed Emami, Saeedeh Noushini, Negar Mohammadhosseini, Nayyereh Shirkavand, Sussan Kabudanian Ardestani, Maliheh Safavi, Marjaneh Samadizadeh, Aida Letafat, Abbas Shafiee, Alireza Foroumadi
Iranian Journal of Basic Medical Sciences, Year. 2013,
Download
162.

Synthesis and Evaluation of Anti-acetylcholinesterase Activity of 2-(2-(4-(2-Oxo-2-phenylethyl)piperazin-1-yl) ethyl)Isoindoline-1,3-dione Derivatives with Potential AntiAlzheimer Effects


Authors: Alireza Aliabadi, Alireza Foroumadi, Ahmad Mohammadi-Farani, Mahdi Garmsiri Mahvar.
Iranian Journal of Basic Medical Sciences, Year. 2013,
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163.

Synthesis,Cytotoxicity Assessment, and Molecular Docking of 4-Substituted-2-p-tolylthiazole Derivatives as Probable c-Src and erb Tyrosine Kinase Inhibitors.


Authors: Alireza Aliabadi, Alireza Foroumadi, Maliheh Safavi, and Sussan K. Ardestani. Synthesis,
Croatica Chemica Acta, Year. 2013,
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164.

Anti-Helicobacter pylori activity and Structure-Activity Relationship study of 2-Alkylthio-5-(nitroaryl)-1,3,4-thiadiazole Derivatives


Authors: Ali Asadipour, Najmeh Edraki, Maryam Nakhjiri, Azadeh Yahya-Meymandi, Eskandar Alipour, Parastoo Saniee, Farideh Siavoshi, Abbas Shafiee and Alireza Foroumadi.
Iranian Journal of Pharmaceutical Research, Year. 2013,
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165.

Quantitative Structure - Activity Relationships Study of Carbonic Anhydrase Inhibitors Using Logistic Regression Model


Authors: Hassan Sahebjamee, Parichehre Yaghmaei, Parviz Abdolmaleki, Alireza Foroumadi
Iranian Journal of Chemistry & Chemical Engineering, , Year. 2013,
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166.

Synthesis and investigation of antioxidant activities of 2-benzylidene-3-coumaranones.


Authors: Hadi Adibi, Alireza Foroumadi, Reza Khodarahmi, Karim Najafi, Mostafa RezaeiTavirani
Journal of Paramedical Sciences , Year. 2013,
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167.

Design, synthesis, biological evaluation and docking study of 5-oxo-4,5-dihydropyrano[3,2-c]chromene derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors


Authors: Mehdi Khoobi, Masoumeh Alipour, Amirhossein Sakhteman, Hamid Nadri, Alireza Moradi, Mehdi Ghandi, Saeed Emami, Alireza Foroumadi, Abbas Shafiee.
European Journal of Medicinal Chemistry, Year. 2013,
168.

Mannich bases of 7-piperazinylquinolones and kojic acid derivatives: Synthesis, in vitro antibacterial activity and in silico study.


Authors: Saeed Emami, Ebrahim Ghafouri, Mohammad Ali Faramarzi, Nasrin Samadi, Hamid Irannejad, Alireza Foroumadi.
European Journal of Medicinal Chemistry, Year. 2013,
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169.

Polyoxygenated cinnamoylcoumarins as conformationally constrained analogs of cytotoxic diarylpentanoids: Synthesis and biological activity.


Authors: Fatemeh Molaverdi, Mehdi Khoobi, Saeed Emami, Masoumeh Alipour, Omidreza Firuzi, Alireza Foroumadi, Gholamreza Dehghan, Ramin Miri, Fatemeh Shaki, Farnaz Jafarpour, Abbas Shafiee.
European Journal of Medicinal Chemistry, Year. 2013,
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170.

Synthesis and psychobiological evaluation of modafinil analogs in mice.


Authors: Arezou Lari, Isaac Karim, Hadi Adibi, Alireza Aliabadi, Loghman Firoozpour, Alireza Foroumadi.
DARU Journal of Pharmaceutical Sciences, Year. 2013,
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171.

Synthesis and biological evaluation of novel benzyl piperazine derivatives of 5-(5-nitroaryl)1,3,4-thiadiazoles as Anti-Helicobacter pylori agents.


Authors: Negar Mohammadhosseini, Parastoo Saniee, Ameneh Ghamaripour, Hassan Aryapour, Farzaneh Afshar, Najmeh Edraki, Farideh Siavoshi, Alireza Foroumadi, Abbas Shafie
DARU Journal of Pharmaceutical Sciences,, Year. 2013,
Download
172.

Synthesis and In vitro cytotoxic activity evaluation of (E)-16-(substituted benzylidene) derivatives of dehydroepiandrosterone.


Authors: Mohsen Vosooghi. Hoda Yahyavi, Kouros Divsalar, Hashem Shamsa, Asma Kheirollahi, Maliheh Safavi, Sussan Kabudanian Ardestani, Sareh Sadeghi-Neshat, Negar Mohammadhosseini, Najmeh Edraki, Mehdi Khoshneviszadeh, Abbas Shafiee and Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences, Year. 2013,
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173.

Synthesis and cytotoxic properties of novel (E)-3-benzylidene-7-methoxychroman-4-one derivatives


Authors: Saeedeh Noushini, Eskandar Alipour, Saeed Emami, Maliheh Safavi, Sussan Kabudanian Ardestani, Ahmad Reza Gohari, Abbas Shafiee and Alireza Foroumadi.
DARU Journal of Pharmaceutical Sciences, Vol.21, No.31, Year. 2013,
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174.

Determination of the role of calcium on instability of neurotoxic metabolite of ecstasy by HPTLC-mass.


Authors: Bardia Jamali, Yalda Hosseinzadeh Ardakani, Mohammad-Reza Rouini, Alireza Foroumadi, Salimeh Amidi, Vahid Hossein Zadeh Aghdam, and Farzad Kobarfard.
DARU Journal of Pharmaceutical Sciences, Vol.21, No.9, Year. 2013,
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175.

Synthesis of 7-Substituted Fluoroquinolone Derivatives Contain- ing Triazolidine Dione Moiety and In Vitro Evaluation of their Cytotoxic Effects.


Authors: Hadi Adibi, Leila Hosseinzadeh, Maryam Mahdian, Alireza Foroumadi, Mohammad Ali Zolfigol, Shadpour Mallakpou
Journal of Reports in Pharmaceutical Sciences, Vol.2, Year. 2013,
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176.

Novel coumarin-3-carboxamides bearing N-benzylpiperidine moiety as potent acetylcholinesterase inhibitors


Authors: Ali Asadipour, Masoumeh Alipour, Mona Jafari, Mehdi Khoobi, Saeed Emami, Hamid Nadri, Amirhossein Sakhteman, Alireza Moradi, Vahid Sheibani, Farshad Homayouni Moghadam, Abbas Shafiee, Alireza Foroumadi.
European Journal of Medicinal Chemistry. , Vol.70, Year. 2013,
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177.

Synthesis and biological evaluation of 3-(trimethoxyphenyl)-2(3H)thiazole thiones as combretastatin analogs.


Authors: Mandana Banimustafa, Asma Kheirollahi, Maliheh Safavi, Sussan Kabudanian Ardestani, Hassan Aryapour, Alireza Foroumadi, Saeed Emami.
European Journal of Medicinal Chemistry , Vol.70, Year. 2013,
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178.

7-Piperazinylquinolones with methylene-bridged nitrofuran scaffold as new antibacterial agents


Authors: Saeed Emami•Nima Shahrokhirad, Alireza Foroumadi, Nasrin Samadi, Mohammad Ali Faramarzi,
MEDICINAL CHEMISTR Y RESEARCH, Vol.22, Year. 2013,
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179.

Microwave-assisted synthesis and anticonvulsant activity of 5,6-bisaryl-1,2,4-triazine-3-thiol derivatives


Authors: Hamid Irannejad, Nima Naderi, Roja Qobadi Ghadikolaei, Ali Mazar-Atabaki, Saeed Emami, Alireza Foroumadi, Sakineh Dadashpour, Tina Zafari
MEDICINAL CHEMISTR Y RESEARCH, Year. 2013,
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180.

Anti-Helicobacter pylori activity and Structure-Activity Relationship study of 2-Alkylthio-5-(nitroaryl)-1,3,4-thiadiazole Derivatives


Authors: Ali Asadipour, Najmeh Edraki, Maryam Nakhjiri, Azadeh Yahya-Meymandi, Eskandar Alipour, Parastoo Saniee, Farideh Siavoshi, Abbas Shafiee, and Alireza Foroumadi.
Iranian Journal of Pharmaceutical Researc, Vol.12, No.3, Year. 2013,
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181.

Synthesis of Monospiro-2-amino-4H-pyran Derivatives Catalyzed by Propane-1-sulfonic Acid-Modified Magnetic Hydroxyapatite Nanoparticles


Authors: Leili Jalili-Baleh, Narges Mohammadi, Mehdi Khoobi, Leila Mamani, Alireza Foroumadi, and Abbas Shafiee
Helvetica Chimica Acta, Vol.96, Year. 2013,
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182.

In vitro Immunobiological Studies of Novel 5-(5-nitrofuran-2-yl)-1, 3, 4Thiadiazoles with Piperazinyl-Linked Benzamidine Substituents against


Authors: Farzaneh Rezazadeh Marznaki, Raheleh Shakeri, Sussan Kaboudanian Ardestani, Azar Tahghighi and Alireza Foroumadi
Iran J Allergy Asthma Immunol , Vol.12, Year. 2013,
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183.

Polyoxygenated cinnamoylcoumarins as conformationally constrained analogs of cytotoxic diarylpentanoids: Synthesis and biological activity


Authors: Fatemeh Molaverdi, Mehdi Khoobi, Saeed Emami, Masoumeh Alipour, Omidreza Firuzi, Alireza Foroumadi, Gholamreza Dehghan, Ramin Miri, Fatemeh Shaki, Farnaz Jafarpour, Abbas Shafiee
European Journal of Medicinal Chemistry, Vol.68, Year. 2013, Number of Page:103-110
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184.

Mannich bases of 7-piperazinylquinolones and kojic acid derivatives: Synthesis, in vitro antibacterial activity and in silico study


Authors: Saeed Emami, Ebrahim Ghafouri, Mohammad Ali Faramarzi, Nasrin Samadi, Hamid Irannejad, Alireza Foroumadi.
European Journal of Medicinal Chemistry, Vol.68, Year. 2013,
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185.

Synthetic Communications: An International Journal for Rapid Communication of Synthetic Organic Chemistry.


Authors: . Mohammad Mahdavi, Mehdi Asadi, Mina Saeedi, Maryam Hosseinpour Tehrani, Seyedeh Sara Mirfazli, Abbas Shafiee & Alireza Foroumadi.
Synthetic Communications, Vol.43, Year. 2013, Number of Page:2936–2942
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186.

New 5-(nitroheteroaryl)-1,3,4-thiadiazols containing acyclic amines at C-2: synthesis and SAR study for their antileishmanial activity


Authors: Azar Tahghighi, Saeed Emami, Sepide Razmi, Farzane Rezazade Marznaki, Sussan Kabudanian Ardestani, Siavoush Dastmalchi, Farzad Kobarfard, Abbas Shafiee, and Alireza Foroumadi
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol.28, No.4, Year. 2013,
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187.

Synthesis and investigation of antioxidant activities of 2-benzylidene-3-coumaranones


Authors: Hadi Adibi, Alireza Foroumadi, Reza Khodarahmi, Karim Najafi, Mostafa RezaeiTavirani
Journal of Paramedical Sciences , Vol.4, Year. 2013,
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188.

REACTION OF ISATOIC ANHYDRIDE, AMINE, AND N,N ’-DIALKYL CARBODIIMIDES UNDER SOLVENT-FREE CONDITIONS: NEW AND EFFICIENT SYNTHESIS OF 3-ALKYL-2-(ALKYLAMINO) QUINAZOLIN-4(3H)-ONES


Authors: Mehdi Asadi, Mina Saeedi, Abbas Shafiee, Mostafa Ebrahimi, Parviz Rashidi Ranjbar,
Synthetic Communications, Vol.43, Year. 2013,
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189.

Dicyano(7-methyl-6-oxo-6H-dibenzo[b,d]pyran-9-yl)methanide Salts via a Multicomponent Reaction


Authors: Mehdi Khoobi, Ali Ramazani, Alireza Foroumadi, Ali Souldozi, Katarzyna S ´ lepokura, Tadeusz Lis, Amir Mahyari, Abbas Shafiee, and Sang Woo Joo
Helvetica Chimica Acta, Vol.96, Year. 2013,
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190.

Synthesis and In vitro cytotoxic activity evaluation of (E)-16-(substituted benzylidene) derivatives of dehydroepiandrosterone


Authors: Mohsen Vosooghi, Hoda Yahyavi, Kouros Divsalar, Hashem Shamsa, Asma Kheirollahi, Maliheh Safavi, Susan Kabudanian Ardestani, Sareh Sadeghi-Neshat, Negar Mohammadhosseini, Najmeh Edraki, Mehdi Khoshneviszadeh, Abbas Shafiee and Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences , Vol.21, No.34, Year. 2013,
191.

AC electrokinetic manipulation of selenium nanoparticles for potential nanosensorapplications


Authors: Seyed Reza Mahmoodi, Marzieh Bayati, Somayeh Hosseinirad, Alireza Foroumadi, Seyed Mahdi Rezayat, Kambiz Gilani
Materials Research Bulletin, Vol.48, Year. 2013,
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192.

Synthesis of Isoindolo[2,1-a]quinazoline-5,11-dione Derivatives via the Reductive One-Pot Reaction of N-Substituted 2-Nitrobenzamides and


Authors: Mohammad Mahdavi, Ramin Najafi, Mina Saeedi, Eskandar Alipour, Abbas Shafiee, and Alireza Foroumadi
Helvetica Chimica Acta, Vol.96, Year. 2013,
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193.

In vitro and in vivo evaluation of an in situ gel forming system for the delivery of PEGylated octreotide


Authors: Laleh Erfani Jabarian, Mohammad Reza Rouini, Fatemeh Atyabi, Alireza Foroumadi, Seyed Mahdi Nassiri, Rassoul Dinarvand
European Journal of Pharmaceutical Sciences, Vol.48, Year. 2013,
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194.

5,6-Dimethoxybenzofuran-3-one derivatives: a novel series of dual Acetylcholinesterase/ Butyrylcholinesterase inhibitors bearing benzyl pyridinium moiety


Authors: Hamid Nadri, Morteza Pirali-Hamedani, Alireza Moradi, Amirhossein Sakhteman, Alireza Vahidi, Ali Asadipour, Nouraddin Hosseinzadeh, Mohammad Abdollahi, Abbas Shafiee, Vahid Sheibani, Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences, Vol.21, Year. 2013,
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195.

5-Nitro-heteroarylidene analogs of 2-thiazolylimino-4-thiazolidinones as a novel series of antibacterial agents


Authors: Nouraddin Hosseinzadeh
MEDICINAL CHEMISTR Y RESEARCH, Vol.22, Year. 2013,
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196.

Novel coumarin derivatives bearing N-benzyl pyridinium moiety: Potent and dual binding site acetylcholinesterase inhibitors.


Authors: Masoumeh Alipour, Mehdi Khoobi, Alireza Foroumadi, Hamid Nadri, Alireza Moradi, Amirhossein Sakhteman , Mehdi Ghandi, Abbas Shafiee
Bioorganic & Medicinal Chemistry, Vol.20, Year. 2012,
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197.

4-Aryl-4H-naphthopyrans derivatives: one-pot synthesis, evaluation of Src kinase inhibitory and anti-proliferative activities.


Authors: Ali Rafinejad, Asal Fallah-Tafti, Rakesh Tiwari, Amir Nasrolahi Shirazi, Deendayal Mandal, Abbas Shafiee, Keykavous Parang, Alireza Foroumadi, Tahmineh Akbarzadeh
DARU Journal of Pharmaceutical Sciences, Vol.20, Year. 2012,
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198.

An efficient piecewise linear model for predicting activity of caspase-3 inhibitors.


Authors: Loghman Firoozpour, Khadijeh Sadatnezhad, Sholeh Dehghani, Eslam Pourbasheer, Alireza Foroumadi, Abbas Shafiee, Massoud Amanlou
DARU Journal of Pharmaceutical Sciences, Vol.20, Year. 2012, Page:31,
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199.

A new strategy based on pharmacophore-based virtual screening in adenosine deaminase inhibitors detection and in-vitro study.


Authors: Roya Bazl, Mohammad Reza Ganjali, Massoud Amanlou, Ali-akbar Saboury, Alireza Foroumadi, Parviz Nourozi.
DARU Journal of Pharmaceutical Sciences, Vol.20, Year. 2012, Page::64,
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200.

QSAR Study of 4-Aryl-4H-Chromenes as a New Series of Apoptosis Inducers Using Different Chemometric Tools


Authors: Mehdi Khoshneviszadeh, Najmeh Edraki, Ramin Miri, Alireza Foroumadi and Bahram Hemmateenejad.
Chemical Biology & Drug Design., Vol.79, Year. 2012, Number of Page:442–458
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201.

One-Pot, Four-Component Synthesis of Novel Imidazo[2,1-b]thiazol-5-amine Derivatives.


Authors: Mohammad Mahdavi, Mehdi Asadi, Mina Saeedi, Mostafa Ebrahimi, Mohammad A. Rasouli, Parviz R. Ranjbar, Alireza Foroumadi, Abbas Shafiee
SYNTHESIS, Vol.44, Year. 2012, Page:3649–3654,
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202.

Crew cut, flower-like and mixed-shaggy micelles prepared from HLH and LHL triblocks as carriers: a comparative study of encapsulation, stability and release properties.


Authors: Salman Hassanzadeh, Sepideh Khoee, Mohamad Mahdavi, Alireza Foroumadi.
Journal of Polymer Research, Vol.19, Year. 2012, Number of Page:9978
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203.

Synthesis of Isoindolo[2,1-a]quinazoline-5,11-dione Derivatives via the Reductive One-Pot Reaction of N-Substituted 2-Nitrobenzamides and


Authors: Mohammad Mahdavi, Ramin Najafi, Mina Saeedi, Eskandar Alipour, Abbas Shafiee, and Alireza Foroumadi
Helvetica Chimica Acta, Vol.96, Year. 2013,
Download
204.

AC electrokinetic manipulation of selenium nanoparticles for potential nanosensorapplications


Authors: Seyed Reza Mahmoodi, Marzieh Bayati, Somayeh Hosseinirad, Alireza Foroumadi, SeyedMahdiRezayat, Kambiz Gilani
Materials Research Bulletin, Vol.21, Year. 2012,
Download
205.

Synthesis and antibacterial activity of novel levofloxacin derivatives containing a substituted thienylethyl moiety


Authors: Negar Mohammadhosseini, Zahra Alipanahi, Eskandar Alipour, Saeed Emami, Mohammad Ali Faramarzi, Nasrin Samadi, Nika Khoshnevis, Abbass Shafiee, and Alireza Foroumadi
DARU Journal of Pharmaceutical Sciences, Vol.20, No.16, Year. 2012,
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206.

Induction of apoptosis through tubulin inhibition in human cancer cells by new chromene-based chalcones


Authors: Hassan Aryapour, Gholam Hossein Riazi, Shahin Ahmadian, Alireza Foroumadi, Majid Mahdavi, and Saeed Emami
Pharmaceutical Biology, Vol.50, No.12, Year. 2012, Number of Page:1551–1560
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207.

Derivative Spectrophotometric Method for Simultaneous Determination of Nickel(II) and Copper(II) Using 6-(Anthracen-2-yl)-2,3-dihydro-1,2,4-triazine-3-thione


Authors: M. BARAZANDEH TEHRANI, S.M.S. MIRKAMALI, E. SOURI and A. FOROUMADI
Asian Journal of Chemistry;, Vol.24, No.6, Year. 2012, Number of Page:4517-4521
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208.

Synthesis and Characterization of 1,10-Phenanthroline-2,9-


Authors: SAMIRA SHABAAN,BAHRAM LETAFAT, NASIM ESMATI, ABBAS SHAFIEE, and ALIREZA FOROUMADI
Asian Journal of Chemistry , Vol.24, No.6, Year. 2012, Number of Page:2819-2820
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209.

Cytotoxic Activity Evaluation and QSAR Study of Chromene-based Chalcones


Authors: Loghman Firoozpour, Najmeh Edraki, Maryam Nakhjiri, Saeed Emami, Maliheh Safavi, Sussan Kabudanian Ardestani, Mehdi Khoshneviszadeh, Abbas Shafiee, and Alireza Foroumadi
Arch Pharm Res, Vol.35, No.12, Year. 2012, Number of Page:2117-2125
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210.

A Clean Synthesis of Novel 3-Alkoxy-2-(benzofuran-3-yl)benzofurans via a One-pot Pseudo Three-component Reaction using H3PW12O40• xH2O as a Catalyst


Authors: Leili Jalili-Baleh, Mehdi Khoobi, Abbas Shafiee, and Alireza Foroumadi
Z. Naturforsch, Vol.67, Year. 2012, Number of Page:165 – 170;
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211.

A green one-pot synthesis of N-alkyl-2-(2-oxoazepan-1-yl)-2-arylacetamide derivatives via an Ugi four-center, three-component reaction in water


Authors: Mohammad Ali Rasouli, Mohammad Mahdavi, Parviz Rashidi Ranjbar, Mina Saeedi, Alireza Foroumadi, Abbas Shafiee
Tetrahedron Letters, Vol.53, Year. 2012, Number of Page:7088–7092
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212.

Synthesis of 2,3-diaryl-5H-imidazo[2,1-a]isoindol-5-ones via the one-pot reaction of 1,2-diketones, 2-formylbenzoic acids, and ammonium acetate


Authors: Maryam Sadat Hosseini-Zare, Mohammad Mahdavi, Mina Saeedi, Mehdi Asadi, Shahrzad Javanshir, Abbas Shafiee, Alireza Foroumadi
Tetrahedron Letters, Vol.53, Year. 2012, Number of Page:3448–3451
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213.

Synthesis of functionalized furo[3,2-c]coumarins via a one-pot oxidative pseudo three-component reaction in poly(ethylene glycol)


Authors: Zeinab Zareai, Mehdi Khoobi, Ali Ramazani, Alireza Foroumadi, Katarzyna Slepokura, Tadeusz Lis, Abbas Shafiee, Ali Souldozi
Tetrahedron, Vol.68, Year. 2012, Number of Page:6721-6726
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214.

Synthesis of Novel 1,4-Benzodiazepine-3,5-dione Derivatives: Reaction of 2-Aminobenzamides under Bargellini Reaction Conditions


Authors: Mohammad Mahdavi, Mehdi Asadi, Mina Saeedi, Zahra Rezaei, Hooman Moghbel, Abbas Shafiee, Alireza Foroumadi
Synlett, Vol.23, Year. 2012, Number of Page:2521–2525
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215.

Antiproliferative Activity of Flavonoids:Influence of the Sequential Methoxylation State of the Flavonoid Structure


Authors: Ghazaal Moghaddam, Soltan Ahmad Ebrahimi, Nahid Rahbar-Roshandel and Alireza Foroumadi
PHYTOTHERAPY RESEARCH, Vol.26, Year. 2012, Number of Page:1023–1028 (2012)
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216.

Synthesis and evaluation of some novel methylene-bridged aryl semicarbazones as potential anticonvulsant agents


Authors: Saeed Mozaffari, Mohsen Amini, Saeed Ghasemi, Hoda Baher, Amirhossein Sakhteman, Abdolrasoul H. Ebrahimabadi , Hamidreza Khademi, Alireza Foroumadi, Mohammad Sharifzadeh
MEDICINAL CHEMISTRY RESEARCH, Vol.21, Year. 2012, Number of Page:3797-3808
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217.

Effects of silica nanoparticles supported ionic liquid as additive on thermal reversibility of human carbonic anhydrase II


Authors: Azadeh Fallah-Bagheri, Ali Akbar Saboury, Leila Ma’mani, Mohammad Taghizadeh,Reza Khodarahmi, Samira Ranjbar, Mousa Bohlooli, Abbas Shafiee, Alireza Foroumadi, Nader
InternationalJournalofBiologicalMacromolecules, Vol.51, Year. 2012, Page:933-938,
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218.

PEGylation of Octreotide Using an α,β-unsaturated-β′-mono-sulfone Functionalized PEG Reagent


Authors: Laleh Erfani-Jabarian, Rasoul Dinarvand, Mohammad Reza Rouini, Fatemeh Atyabi, Mohsen Amini, Negar Mohammadhosseini, Abbas Shafiee, and Alireza Foroumadi
Iranian Journal of Pharmaceutical Research, Vol.11, No.3, Year. 2012, Number of Page:747-753
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219.

Highly cis-Diastereoselective Synthesis of Coumarin-Based 2,3-Disubstituted Dihydrobenzothiazines by Organocatalysis


Authors: Mehdi Khoobi, Ali Ramazani, Alireza Foroumadi, Saeed Emami, Farnaz Jafarpour, Amir Mahyari, Katarzyna S lepokura, Tadeusz Lis, and Abbas Shafiee
Helvetica Chimica Acta, Vol.95, Year. 2012, Page:660-671,
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220.

Cell death features induced in Leishmania major by 1,3,4-thiadiazole derivatives


Authors: Sussan K. Ardestani, Fatemeh Poorrajab, Sepideh Razmi, Alireza Foroumadi, Behnaz Gharegozlou, Mina Behrouzi-Fardmoghadam, Abbas Shafiee, Soheila Ajdary
Experimental Parasitology, Vol.132, Year. 2012, Number of Page:116–122
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221.

Halogenated flavanones as potential apoptosis-inducing agents: Synthesis and biological activity evaluation


Authors: Maliheh Safavi, Nasim Esmati, Sussan Kabudanian Ardestani, Saeed Emami, Jamshid Davoodi, Abbas Shafiee, Alireza Foroumadi, Soheila Ajdari
European Journal of Medicinal Chemistry 58, Vol.58, Year. 2012, Number of Page:573-580
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222.

Replacement of the Methylene of Dihydrochalcones with Oxygen: Synthesis and Biological Evaluation of 2-Phenoxyacetophenones


Authors: Mahsa Ansari, Saeed Emami, Mohammad A. Khalilzadeh, Malek T. Maghsoodlou, Alireza Foroumadi, Mohammad A. Faramarzi and Sussan K. Ardestani, Nasrin Samadi
Chem Biol Drug Des 2012;, Vol.80, Year. 2012, Number of Page:591–597
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223.

2-Amino-3-cyano-4-(5-arylisoxazol-3-yl)-4H-chromenes: Synthesis and In Vitro Cytotoxic Activity


Authors: Tahmineh Akbarzadeh, Ali Rafinejad, Javad Malekian Mollaghasem, Maliheh Safavi, Asal Fallah-Tafti, Mahboobeh Pordeli, Sussan Kabudanian Ardestani, and Alireza Foroumadi, Abbas Shafiee
Archive dre pharmazie, Vol.345, Year. 2012, Number of Page:386–392
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224.

Anti-proliferative and Apoptotic Effects of the Derivatives from 4aryl-4H-chromene Family on Human Leukemia K562 Cells


Authors: Hassan Aryapour, Majid Mahdavi, Seyed Reza Mohebbi, Mohammad Reza Zali, and Alireza Foroumadi
Archives of Pharmacal Research , Vol.35, No.9, Year. 2012, Number of Page:1573-1582
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225.

Anti-Helicobacter pylori Activity of the Methanolic Extract of Geum iranicum and its Main Compounds


Authors: Somayeh Shahani, Hamid R.Monsef-Esfahani, Soodabeh Saeidnia, Parastoo Saniee, Farideh Siavoshi, Alireza Foroumadi, Nasrin Samadi, and Ahmad R. Gohari
Z. Naturforsch., Vol. 67, Year. 2012, Number of Page:172 – 180
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226.

Bis(dicyclohexylaminium) 2-carboxymethyl-2-hydroxysuccinate ethanol monosolvate


Authors: Mahsa Foroughian,Hossein Aghabozorg, Behrouz Notash, Abbas Shafiee,and Alireza Foroumadi
Acta Crystallographica Section E, Vol.68, Year. 2012, Number of Page:o2792–o2793
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227.

Safety and Ef?cacy of New 3,6-diaryl-7H[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine Analogs as Potential Phosphodiesterase-4 Inhibitors in NIH3T3 Mouse Fibroblastic Cells


Authors: Maryam Baeeri, Alireza Foroumadi, Maryam Motamedi, Azadeh YahyaMeymandi, Loghman Firoozpour, Seyed N. Ostad, Abbas Shafiee, Saeid Souzangarzadeh and Mohammad Abdollahi
Chemical Biology & Drug Design, Vol.78, Year. 2011, Page:444-438,
228.

.1-[(2-Arylthiazol-4-yl)methyl]azoles as a New Class of Anticonvulsants: Design, Synthesis, In vivo Screening, and In silico Drug-like Properties


Authors: Nematollah Ahangar, Adile Ayati, Eskandar Alipour, Arsalan Pashapour, Alireza Foroumadi , Saeed Emami
Chemical Biology & Drug Design, Vol.78, Year. 2011, Page:852-844,
229.

Synthesis and Free Radical Scavenging Activity of Coumarin Derivatives Containing a 2-Methylbenzothiazoline Motif


Authors: Mehdi Khoobi, Saeed Emami, Gholamreza Dehghan, Alireza Foroumadi, Ali Ramazani, Abbas Shafiee
Arch. Pharm. Chem. Life Sci, Vol.344, Year. 2011, Page:594-588,
230.

3-Diaminopyridinium 6-carboxypyridine-2-carboxylate


Authors: Mahsa Foroughian, Alireza Foroumadi, Behrouz Notash,Giuseppe Bruno, Hadi Amiri Rudbari Hossein Aghabozorg
Acta Cryst, No.67, Year. 2011, Page:o3325,
231.

Concomitant activation of caspase-9 and down-regulation of IAP proteins as a mechanism of apoptotic death in HepG2, T47D and HCT-116 cells upon exposure to a derivative from 4-aryl-4H-chromenes family


Authors: Majid Mahdavi, Jamshid Davoodi, Mohammad Reza Zali, Alireza Foroumadi
Biomedicine & Pharmacotherapy , Vol.65, Year. 2011, Page:182-175,
232.

Optimization of the simultaneous determination of imatinib and its major metabolite, CGP74588, in human plasma by a rapid HPLC method using D-optimal experimental design


Authors: Ali-Akbar Golabchifar, Mohammad-Reza Rouini, Bijan Shafaghi, Alireza Foroumadi, Mohammad-Reza, Khoshayand, Saeed Rezaee
Talanta , Vol.85, Year. 2011, Page:2329-2320,
233.

4-Aryl-4H-Chromene-3-Carbonitrile Derivatives: Evaluation of Src Kinase Inhibitory and Anticancer Activities


Authors: Asal Fallah-Tafti, Rakesh Tiwari, Amir Nasrolahi Shirazi, Tahmineh Akbarzadeh, Deendayal Mandal, Abbas Shafiee, Keykavous Parang, Alireza Foroumadi
Medicinal Chemistry, Vol.7, Year. 2011, Page:472-466,
234.

Efficient Microwave-Assisted Synthesis of 3-Benzothiazolo and 3-Benzothiazolino Coumarin Derivatives Catalyzed by Heteropoly Acids


Authors: M. Khoobi, A. Ramazani, A. Foroumadi, H. Hamadi, Z. Hojjati, and A. Shafiee
J. Iran. Chem. Soc., Vol.8, No.4, Year. 2011, Page:1042-1036,
235.

Thiazolyl N-benzyl-substituted acetamide derivatives: Synthesis, Src kinase inhibitory and anticancer activities


Authors: Asal Fallah-Tafti, Alireza Foroumadi, Rakesh Tiwari, Amir Nasrolahi Shirazi, Yahao Bu, Tahmineh Akbarzadeh, Keykavous Parang, Abbas Sha?ee
European Journal of Medicinal Chemistry, Vol.48, Year. 2011, Page:4858-4853,
236.

eCoumarin-Based Bioactive Compounds: Facile Synthesis and Biological Evaluation of Coumarin-Fused 1,4-Thiazepines


Authors: Mehdi Khoobi, , Alireza Foroumadi, Saeed Emami, Maliheh Safavi, Gholamreza Dehghan, Babak H. Alizadeh, Ali Ramazani, Sussan K. Ardestani. and Abbas Sha?
Chem Biol Drug Des , Vol.78, Year. 2011, Page:586-580,
237.

Synthesis and Antifungal Activity of 1-[(2Benzyloxy)Phenyl]-2-(Azol-1-yl)Ethanone Derivatives: Exploring the Scaffold Flexibility


Authors: Saeed Emami, Motahare KazemiNajafabadi, Soughra Pashangzadeh, Alireza Foroumadi, Mohammad Ali Faramarzi, Nasrin Samadi, Mehraban Falahati, Roohollah Fateh and Mahtab Ashra Khozani
Chem Biol Drug Des , Vol.78, Year. 2011, Page:987-979,
238.

Anti-angiogenic/proliferative behavior of a ‘‘4-aryl-4H-chromene’’ on blood vessel’s endothelial cells: A possible evidence on dual ‘‘anti-tumor’’ activity


Authors: Kamran Mansouri, Reza Khodarahmi, Alireza Foroumadi, Ali Mostafaie, Hamidreza Mohammadi Motlagh
Med Chem Res , Vol.20, Year. 2011, Page:929-920,
239.

In vitro antibacterial activity of some Iranian medicinal plant extracts against Helicobacter pylori


Authors: M. Hajimahmoodi, M. Shams-Ardakani, P. Saniee, F. Siavoshi, M. Mehrabani, H. Hosseinzadeh, P. Foroumadi, M. Safavi, M. Khanavi, T. Akbarzadeh, A. Shafiee, A. Foroumadi
Natural Product Research, Vol.25, No.11, Year. 2011, Page:1066-1059,
240.

Synthesis and In-vitro Antibacterial Activities of Acetylanthracene and Acetylphenanthrene Derivatives of Some Fluoroquinolones


Authors: Fazel Shamsa, Alireza Foroumadi, Hashim Shamsa, Nasrin Samadi, Mohammad Ali Faramarzi, Abbas Shafiee
Iranian Journal of Pharmaceutical Research , Vol.10, No.2, Year. 2011, Page:231-225,
241.

Synthesis and In Vitro Cytotoxic Activity of N-2-(2-Furyl)-2-(chlorobenzyloxyimino) Ethyl Ciprofloxacin Derivatives


Authors: Eskandar Alipour, Negar Mohammad hosseini, Fatemeh Panah, Sussan K.Ardestani, Maliheh Safavi, Abbas Shafiee, Alireza Foroumadi
E-Journal of Chemistry , Vol.8, No.3, Year. 2011, Page:1231-1226,
242.

Synthesis and In Vitro Antibacterial Activity of New 2-(1-Methyl-4-nitro-1H-imidazol-5-ylsulfonyl)-1,3,4-thiadiazoles


Authors: Bahram Letafats, Negar Mohammad Hosseinis, Ali Asadipour, Alireza Foroumadi
E-Journal of Chemistry , Vol.8, No.3, Year. 2011, Page:1123-1120,
243.

Aminopropyl-functionalized cubic Ia3d mesoporous silica nanoparticle as an efficient support for immobilization of superoxide dismutase


Authors: Mojtaba Falahati, Leila Ma'mani, Ali Akbar Saboury, Abbas Shafiee, Alireza Foroumadi, Ali Reza Badiei
Biochimica et Biophysica Acta , Vol.1814, Year. 2011, Page:1202-1195,
244.

Synthesis and Spectroscopic Characterization of New Axially Coordinated Cobalt(III) Schiff Base Complexes


Authors: N. Esmati, M.Yousefi, A.Shafiee, A.Foroumadi
Asian Journal of Chemistry, Vol.23, No.9, Year. 2011, Page:4013-4011,
245.

Synthesis of 1-[3-(Cyclopentyloxy)-4-methoxyphenyl]cyclopentanol as Potential Phospho diesterase-4 Inhibitor


Authors: A. Yahya-Meymandi, G. Mohammadi ziaraniO, A. Shafiee, A. Foroumadi
Asian Journal of Chemistry , Vol.23, No.9, Year. 2011, Page:4010-4008,
246.

Synthesis and anti-Helicobacter pylori activity of (4-nitro-1-imidazolylmethyl)-1,2,4-triazoles, 1,3,4-thiadiazoles, and 1,3,4-oxadiazoles


Authors: Asal Fallah tafti, Tahmineh Akbarzadeh, Parastoo Saniee, Farideh Siavoshi, Abbas Shafiee, Alireza Foroumadi
Turk J Chem , Vol.35, Year. 2011, Page:316-307,
247.

Biological evaluation of synthetic analogues of curcumin: chloro-substituted-20-hydroxychalcones as potential inhibitors of tubulin polymerization and cell proliferation


Authors: Hassan Aryapour, Gholam Hossein Riazi, Alireza Foroumadi, Shahin Ahmadian, Abbas Shafiee, Oveis Karima, Majid Mahdavi, Saeed Emami, Maedeh Sorkhi, Sirus Khodadady
Med Chem Res, Vol.20, Year. 2011, Page:510-503,
248.

Synthesis of Novel 2-(2-Methylsulfonyl-1-methyl-1H-imidazol-5-yl)-5-(alkylsulfonyl)-1,3,4-thiadiazoles


Authors: Azita Javidnia, Tahmineh Akbarzadeh, Loghman Firoozpour, Mehdi Khoobi, Abbas Shafiee, and Alireza Foroumadia
J. Heterocyclic Chem, Vol.48, Year. 2011, Page:457-454,
249.

Synthesis and antileishmanial activity of novel 5-(5-nitrofuran-2-y1)-1,3,4-thiadiazoles with piperazinyl-linked benzamidine substituents


Authors: Azar Tahghighi, Farzane Rezazade Marznaki, Farzad Kobarfard, Siavoush Dastmalchi, Javid Shahbazi Mojarrad, Sepideh Razmi, Sussan Kabudanian Ardestani, Saeed Emami, Abbas Shafiee, Alireza Foroumadi
European Journal of Medicinal Chemistry, Vol.46, Year. 2011, Page:2608-2602,
250.

Synthesis and In Vitro Cytotoxic Activity of 2-Amino-7-(dimethylamino)-4-[(trifluoromethyl)phenyl]-4H-chromenes


Authors: M. Mahdavi, A. Asadipour, S. Rajabalian, M. Vosooghi, L. Firoozpour, M. Nakhjiri, A. Shafiee and A. Foroumadi
E-Journal of Chemistry, Vol.8, No.2, Year. 2011, Page:602-598,
251.

Antinociceptive activity of some 1,4-substituted Piperidine derivatives using tail flick method in mice


Authors: Amirhossein Sakhteman, Mohammad Sharifzadeh, Alireza Moradi, Hamid Nadri, Kaveh Tabrizian, Massoud Amanlou, Ali Asadipour, Kouros Divsalar, Abbas Shafiee and Alireza Foroumadi
African Journal of Pharmacy and Pharmacology, Vol.5, No.3, Year. 2011, Page:357-352,
252.

Giuseppe Bruno and Hadi Amiri Rudbari. N1,N1-Dimethylpropane-1,2-diaminium bis(6-carboxypyridine-2-carboxylate) monohydrate


Authors: Hossein Aghabozorg, Mahsa Foroughian, Alireza Foroumadi
Acta Crystallographica Section , Vol.67, Year. 2011, Page:o932–o933,
253.

Synthesis of 1-Benzyl-4-[2-(5-phenyl-1,3,4-thiadiazole-2-yl)aminoethyl]piperidine as Potential Alzheimer's Disease Modifying Agent


Authors: Diba Nabardi Sarkandi, Loghman Firoozpour, AliAsadipour, Vahid Sheibani, Mahsa Alizadeh Monavar Asli, Asghar Davood, Abbas Shafiee and Alireza Foroumadi
Asian Journal of Chemistry, Vol.23, Year. 2011, Page:2505-2503,
254.

Synthesis of 1-Benzyl-4-[2-(3-thienylcarbonylamino)ethyl]piperidine as a Novel Potential Cholinesterase Inhibitor


Authors: Mahsa Alizadeh Monavar Asli, Loghman Firoozpour, Vahid Sheibani, Diba Nabardi Sarkandi, Amirhossein Sakhteman, Asghar Davood, Abbas Shafiee and Alireza Foroumadi
Asian Journal of Chemistry, Vol.23, Year. 2011, Page:2490-2487,
255.

Synthesis and biological activity of 5-nitrofuran-containing (1,3,4-thiadiazol-2-yl) piperazine moieties as a new type of anti-Helicobacter pylori heterocycles


Authors: Mohammad Hassan Moshafi, Azadeh Yahya- Meymandi, Seyed Esmaeil Sadat-Ebrahimi, Saeeid Emami, Maryam Nakhjiri, Farideh Siavoshi, Maryam Omrani, Mohsen Vosooghi, Eskandar Alipour, Abbas Shafiee and Alireza Foroumadi
J. Serb. Chem. Soc, Vol.76, Year. 2011, Page:210-201,
256.

Synthesis and antileishmanial activity of 5-(5-nitroaryl)-2-substituted-thio-1,3,4-thiadiazoles


Authors: Eskandar Alipour, Saeed Emami, Azadeh Yahya-Meymandi, Maryam Nakhjiri, Farnaz Johari,Sussan K. Ardestani, Fatemeh Poorrajab, Maryam Hosseini, Abbas Shafiee, and Alireza Foroumadi
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol.26, Year. 2011, Page:128-123,
257.

Nanocomposite Based Carbon Paste Electrode for Selective Analysis of Copper


Authors: Mohammad Reza Ganjali, Sajjad Aghabalazadeh, Mehdi khoobi, Ali Ramazani, Alireza Foroumadi, Abbas Shafiee and Parviz Norouzi
Int. J. Electrochem. Sci, Vol.6, Year. 2011, Page:62-52,
258.

5-Nitroimidazole-based 1,3,4-Thiadiazoles: Heterocyclic Analogs of Metronidazole as Anti-Helicobacter pylori Agents


Authors: Mohammad Hassan Moshafi, Maedeh Sorkhi, Saeed Emami, Maryam Nakhjiri, Azadeh Yahya-Meymandi, Amir Soheil Negahbani, Farideh Siavoshi, Maryam Omrani, Eskandar Alipour, Mohsen Vosooghi, Abbas Shafiee, and Alireza Foroumadi
Arch. pharm. Chem. Life Sci, Vol.11, Year. 2011, Page:183-178,
259.

Discovery of a novel nitroimidazolyle oxazolidinone hybrid with potent anti Gram-positive activity: Synthesis and antibacterial evaluation


Authors: Ali Khalaj, Maryam Nakhjiri, Amir Soheil Negahbani, Marjaneh Samadizadeh, Loghman Firoozpour, Saeed Rajabalian, Nasrin Samadi, Mohammad Ali Faramarzi, Neda Adibpour, Abbas Shafiee, Alireza Foroumadi
European Journal of Medicinal Chemistry , Vol.46, Year. 2011, Page:70-65,
260.

Isochaihulactone analogues: Synthesis and anti-proliferative activity of novel dibenzylbutyrolactones


Authors: Babak Heidary Alizadeh, Alireza Foroumadi, Saeed Emami, Mehdi Khoobi, Fatemeh Panah, Sussan K. Ardestani, Abbas Shafiee
European Journal of Medicinal Chemistry, Vol.45, Year. 2011, Page:5979-5984,
261.

Synthesis and cytotoxic activity of some 2-amino-4-aryl-3-cyano-7-(dimethylamino)-4H-chromenes


Authors: M. Vosooghi, S. Rajabalian, M. Sorkhi, M. Badinloo, M. Nakhjiri, A.S. Negahbani,A. Asadipour, M. Mahdavi, A. Shafiee, A. Foroumadi
Research in Pharmaceutical Sciences, Vol.5, No.1, Year. 2010, Page:18-13,
262.

Synthesis and biological evaluation of 2-phenylthiazole-4-carboxamide derivatives as anticancer agents


Authors: Alireza Aliabadi, Fazel Shamsa, Seyed Nasser Ostad, Saeed Emami, Abbas Shafiee, Jamshid Davoodi, Alireza Foroumadi
European Journal of Medicinal Chemistry , Vol.45, Year. 2010, Page:5389-5384,
263.

Heterocycle-bridged and Conformationally Constrained Retinoids: Synthesis of 4-(7,8,9,10-Tetrahydro-7,7,10,10-tetramethyl-4H-benzo[6,7]chromeno-[4,3-d]thiazole-2-yl) benzoic Acid


Authors: Lamei Navid, Foroumadi Alireza, Emami Saeed, Amini Mohsen, Shafiee Abbas
Chinese Journal of chemistry, Vol.28, Year. 2010, Page:1956-1951,
264.

Synthesis of Two Novel 3-Amino-5-[4-chloro-2-phenoxyphenyl]-4H-1,2,4-triazoles with Anticonvulsant Activity


Authors: Mahdavi Mohammad, Akbarzadeh Tahmineh, Sheibani Vahid, Abbasi Maryam, Firoozpour Loghman, Tabatabai Sayyed Abbas, Shafiee Abbas, Foroumadi Alireza
Iranian Journal of Pharmaceutical Research, Vol.9, No.3, Year. 2010, Page:269-265,
265.

Development and validation of a rapid HPLC- fluorescence method for simultaneous determination of venlafaxine and its major metabolites in human plasma


Authors: Ardakani, Y. H., Foroumadi, A., Rouini, M. R
Daru-Journal of Faculty of Pharmacy , Vol.18, No.2, Year. 2010, Page:102-97,
266.

Synthesis and cloxacillin antimicrobial enhancement of 2-methylsulfonylimidazolyl-1,4-dihydropyridine derivatives


Authors: Akbarzadeh, T, Tafti, Fallah A., Samadi, N., Foroumadi, A., Amanlou, M., Faramarzi, M. A., Shafiee, A
Daru-Journal of Faculty of Pharmacy, Vol.18, No.2, Year. 2010, Page:123-118,
267.

Design, synthesis and anticholinesterase activity of a novel series of 1-benzyl-4-((6-alkoxy-3-oxobenzofuran-2(3H)-ylidene) methyl) pyridinium derivatives


Authors: Hamid Nadri, Morteza Pirali-Hamedani, Maryam Shekarchi, Mohammad Abdollahi, Vahid Sheibani, Massoud Amanlou, Abbas Shafiee and Alireza Foroumadi
Bioorganic & Medicinal Chemistry, Vol.18, No.17, Year. 2010, Page:6366-6360,
268.

Synthesis and in-vitro Cytotoxicity of Poly-functionalized 4-(2-Arylthiazol-4-y1)-4H-chromenes


Authors: Mahmoodi, Majid, Aliabadi, Alireza, Emami, Saeed, Safavi, Maliheh, (Rajabalian, Saeed, Mohagheghi, Mohammad-Ali, Khoshzaban, Ahad, Samzadeh-Kermani, Alireza, Lamei, Navid, Shafiee, Abbas, Foroumadi, Alireza
Archiv der Pharmazie, Vol.343, No.7, Year. 2010, Page:416-411,
269.

Chromene-Based Synthetic Chalcones as Potent Antileishmanial Agents: Synthesis and Biological Activity


Authors: Alireza Foroumadi, Saeed Emami, Maedeh Sorkhi, Maryam Nakhjiri, Zohreh Nazarian, Samaneh Heydari, Sussan K. Ardestani, Fatemeh Poorrajab, Abbas Shafiee
Chemical Biology & Drug Design, Vol.75, No.10, Year. 2010, Page:596-590,
270.

Complexes of 2-hydroxyacetophenone semicarbazones: A novel series of superoxide dismutase mimetics


Authors: Maliheh Safavi, Alireza Foroumadi, Maryam Nakhjiri, Mohammad Abdollahi, Abbas Shafiee, Hoda Ilkhani, Mohammad Reza Ganjali, Seyed Jalal Hosseinimehr and Saeed Emami
Bioorganic & Medicinal Chemistry Letters, Vol.20, No.10, Year. 2010, Page:3073-3070,
271.

Comparative studies of mercapto thiadiazoles self-assembled on gold nanoparticle as ionophores for Cu(II) carbon paste sensors


Authors: Mohammad Hossein Mashhadizadeh, Hadi Khani, Alireza Foroumadi and Parishad Sagharichi
Analytica Chimica Acta, Vol.665, No.2, Year. 2010, Page:214-208,
272.

Novel antileishmanial chalconoids: Synthesis and biological activity of 1- or 3-(6-chloro-2H-chromen-3-yl)propen-1-ones


Authors: Zohreh Nazarian, Saeed Emami, Samaneh Heydari, Sussan K. Ardestani, Maryam Nakhjiri, Fatemeh Poorrajab, Abbas Shafiee and Alireza Foroumadi
European Journal of Medicinal Chemistry, Vol.45, No.4, Year. 2010, Page:1429-1424,
273.

In vitro cytotoxicity and apoptotic inducing activity of the synthesized 4-aryl-4H-chromenes derivatives against human cancer cell lines


Authors: Mahmoodi M, Rajabalian S, Foroumadi A, Hidarykeshel S, Safavi M, Khoshzaban A, Divsalar K, Mohagheghi MA
Tehran University Medical Journal, Vol.67, No.6, Year. 2009, Page:392-387,
274.

In Vitro Susceptibility of the gram-negative bacterium Helicobacter Pylori to Extracts of Iranin medicinal plants


Authors: Manijeh Atapour, Mohammad Javad Zahedi, Mitra Mehrabani, Maliheh safavi, Vahid Keyvanfard, Akram Foroughi, Farideh Siavoshi, and Alireza Foroumadi
Pharmaceutical Biology, Vol.47, No.1, Year. 2009, Page:80-77,
275.

Evaluation of Anti-inflammatory and Analgesic Activity of a Novel Rigid 3,4-Dihydroxy Chalcone in Mice


Authors: M. R. Heidari, A. Foroumadi, A. Amirabadi, A. Samzadeh-Kermani, B.S. Azimzadeh,and A. Eskandarizadeh
Ann.Acad.Sci, Vol.1171, Year. 2009, Page:406-399,
276.

3-Imidazolyl-Substituted Flavans as Potential Antifungal Agents: Synthesis, Stereochemical Properties, and Antifungal Activity


Authors: Saeed Emami and Alireza Foroumadi
Arch. Pharm. Chem. Life Sci, Vol.342, Year. 2009, Page:545-541,
277.

Synthesis and dopaminergic activity of some E-3-(piperidin-1-yl)-1-(4-substituted phenyl)prop-2-en-1-one derivatives


Authors: Amirhossein Sakhteman, Alireza Foroumadi, Mohammad Sharifzadeh, Masoud Amanlou,Farhoud Rayatnia, Abbas Shafiee
Bioorganic & Medicinal Chemistry , Vol.17, Year. 2009, Page:6913-6908,
278.

Design of Conformationally Constrained Azole Antifungals: Efficient Synthesis and Antifungal Activity of trans-3-Imidazolylflavanones


Authors: Saeed Emami, Mehran Behdad, Alireza Foroumadi, Mehraban Falahati, Ensieh Lotfali and Somaye Sharifynia
Chem Biol Drug Des, Vol.73, Year. 2009, Page:395-388,
279.

Synthesis and Structure-Activity Relationship Study of 2-Substituted- 5-(5-nitro-2-thienyl)-1,3,4-thiadiazoles as Anti-Helicobacter pylori Agents


Authors: Alireza Foroumadi, Somayeh Sedaghat, Saeed Emami, Maryam Yazdanian, Mohammad Hassan Moshafi, Maliheh Safavi1, Amirhossein Sakhteman, Loghman Firoozpour, Mohsen Vosooghi1 and Abbas Shafiee
Letters in Drug Design & Discovery, Vol.6, Year. 2009, Page:474-468,
280.

Study of the anti-Inflammatory and Analgesic effects of Novel Rigid Benzofuran-3,4-diHydroxy Chalcone by Formalin, Hot Plate and Carrageenan tests in Mice. Pak


Authors: Mahmoud Reza Heidari, Alireza Foroumadi,Hojat Noroozi,Ali Samzadeh-Kermani,and Behzad Sarvar Azimzadeh
J. Pharm. Sci, Vol.22, No.4, Year. 2009, Page:401-395,
281.

Synthesis and in vitro anti-Helicobacter pylori activity of 2-(substituted benzylthio)-5-(5-nitro-2- furyl)-1, 3,4-thiadiazole derivatives


Authors: Negar Mohamadhosseini,AliAsadipour, Bahram Letafat,Mohsen Vosoghi, Farideh SIAVOSHI, Abbas Shafiee, Alireza Foroumadi
Turk J Chem, Vol.33, Year. 2009, Page:478-471,
282.

Sensitive Quantification of Carboxylic Acid Metabolite of Clopidogrel in Human Plasma by LC With UV Detection


Authors: Mohammad-Reza.Rouini,Yalda H.Ardakani, Alireza Foroumadi, Hada Lavasani, Lida Hakemi
Choromatographia , Vol.70, No.6/5, Year. 2009,
283.

Synthesis and Structure-Activity Relationship Study of 2-Substituyed-5-(5-nitro-2-thienyl)-1,3,4-thiadiazoles as Anti-Helicobacter Pylori Agents


Authors: Alireza Foroumadi,Somayeh Sedaghat,Saeed Emami, Maryam Yazdanian, Mohammad Hassan Moshafi, Maliheh Safavi, AQmirhossein Sakhteman, Loghman Firoozpour, Mohsen Vosooghi and Abbas Shafiee
Letter Drug Descovery, Vol.6, Year. 2009, Page:474-468,
284.

One-Pot Synthesis of 4-Hydroxy-3-phenyl-2Hpyrano[3,2-b]benzofuran-2-one Derivatives


Authors: Foroumadi A, Zamanian S, Samzadeh-Kermani A, Shafiee A
Synthetic Communications, Vol.39, Year. 2009, Page:1728-1722,
285.

N-Substituted piperazinyl quinolones as potential cytotoxic agents: Structureeactivity relationships study


Authors: Foroumadi, A., Emami, S., Rajabalian, S., Badinloo, M., Mohammadhosseini, N., Shafiee, A
Biomedicine & Pharmacotherapy, Vol.63, Year. 2009, Page:220-216,
286.

Conformationally Constrained Analogs of N-Substituted Piperazinylquinolones: Synthesis and Antibacterial Activity of N-(2,3-Dihydro-4-hydroxyimino-4H-1-benzopyran-3-yl)- piperazinylquinolones


Authors: Saeed Emami, Alireza Foroumadi, Nasrin Samadi, Mohammad A. Faramarzi,and Saeed Rajabalian
Arch. Pharm. Chem. Life Sci, Vol.342, Year. 2009, Page:411-405,
287.

Faramarzie and A. Foroumadi. Synthesis and Antibacterial Activity of N-[2-(2-naphthyl)ethyl]piperazinyl Quinolones


Authors: A. Shafiee, S. Emamic, S. Ghodsid, S. Najjaria, M. Sorkhia, N. Samadie, M.A
J. Iran. Chem. Soc, Vol.6, No.2, Year. 2009, Page:333-325,
288.

Synthesis and Leishmanicidal Evaluation of Novel 4- Substituted-2,2-Dimethyl-7-(prop-2-ynyloxy)Chromenes


Authors: Alizadeh BH , Foroumadi A, Ardestani SK, Poorrajab F, Shafiee A
Turk J Chem, Vol.33, Year. 2009, Page:58-47,
289.

Design of Conformationally Constrained Azole Antifungals: Efficient Synthesis and Antifungal Activity of trans-3-Imidazolylflavanones


Authors: Emami S, Behdad M, Foroumadi A, Falahati M, Lotfali E, Sharifynia S
Chem. Biol. Drug Des, Vol.73, Year. 2009, Page:395-388,
290.

Selective leishmanicidal effect of 1,3,4-thiadiazolederivatives and possible mechanism of action against Leishmania specie


Authors: Poorrajab F., Ardestani S. K., Foroumadi A., Emami S., Kariminia A., Behrouzi,Fardmoghadam M., Shafiee A
Experimental Parasitology , Vol.121, Year. 2009, Page:330-323,
291.

Nitroimidazolyl-1,3,4-thiadiazole-based anti-leishmanial agents: Synthesis and in vitro biological evaluation


Authors: Poorrajab, F., Ardestani, S. K., Emami, S., Behrouzi-Fardmoghadam, M., Shafiee, A., Foroumadi, A
European Journal of Medicinal Chemistry, Vol.44, Year. 2009, Page:1762-1758,
292.

Synthesis and antibacterial activity of nitroaryl thiadiazole-gatifloxacin hybrids


Authors: Jazayeri S., Moshafi M.H., Firoozpour L., Emami S., Haddad M., Pahlavanzadeh F., Esnaashari M., A. Shafiee , Foroumadi A
European Journal of Medicinal Chemistry, Vol.44, Year. 2009, Page:1209-1205,
293.

In vitro susceptibility of gram-negative bacteria helicobacter pylori to extracts of Iranian medicinal plants


Authors: Atapour, M., Zahedi, M. J., Mehrabani, M., Safavi, M., Keyvanfard, V., Foroughi, A., Siavoshi, F., Foroumadi, A
Pharmaceutical Biology , Vol.47, Year. 2009, Page:80-77,
294.

A Convenient Method for the Preparation of Losartan Active Metabolite (EXP-3174)


Authors: Morteza Pirali-Hamedani, Alireza Aliabadi, M. Shekarchi, M. Amini,Mohammad reza rouini, Abbas Shafiee and Alireza Foroumadi.
Asian Journal of Chemistry, Vol.21, No.6, Year. 2009, Page:4913-4909,
295.

Synthesis and anti-Helicobacter pylori activity of 5-(nitroaryl)-1,3,4-thiadiazoles with certain sulfur containing alkyl side chain


Authors: Foroumadi, A., Rineh, A., Emami, S., Siavoshi, F., Massarrat, S., Safari, F., Rajabalian, S., Falahati, M., Lotfalif, E., Shafieea, A
Bioorganic & Medicinal Chemistry Letters, Vol.18, Year. 2008, Page:3320-3315,
296.

Synthesis and in vitro anti-leishmanial activity of [5-(5-nitrofuran-2-yl)-1,3,4-thiadiazol-2-yl]- and 1-[5-(5-nitrothiophen-2-yl)-1,3,4-thiadiazol-2-yl]-4-aroylpiperazin


Authors: Behrouzi-Fardmoghadam, M., Poorrajab, F., Kaboudanian Ardestani, S., Emami, S., Shafiee, A., Foroumadi, A
Bioorganic & Medicinal Chemistry, Vol.16, Year. 2008, Page:4515-4509,
297.

2-Hydroxyphenacyl azoles and related azolium derivatives as antifungal agents


Authors: Emami, S., Foroumadi, A., Falahati, M., Lotfali, E., Rajabalian, S., Ebrahimi, AS., Farahyar, S., Shafiee, A
Bioorganic & Medicinal Chemistry Letters, Vol.18, Year. 2008, Page:146-141,
298.

Synthesis and in vitro anti-Helicobacter pylori activity of N-[5-(5-nitro-2-heteroaryl)-1,3,4-thiadiazol-2-yl]thiomorpholines and related compounds


Authors: Mirzaei J, Siavoshi F, Emami S, Safari F, Khoshayand MR, Shafiee A, Foroumadi A
European Journal of Medicinal Chemistry , Vol.43, No.8, Year. 2008, Page:1580-1575,
299.

Leishmanicidal Evaluation of Novel Synthetic Chromenes Arch


Authors: Alizadeh B. H., Foroumadi A., Ardestani S. K., Poorrajab F., Shafiee A
Pharm. Chem. Life Sci, Vol.341, Year. 2008, Page:793-787,
300.

Effects of novel antituberculosis agents on OmpF channel activity


Authors: Mahdiuni H, Mobasheri H, Shafiee A, Foroumadi A
Biochem Biophys Res Commun, Vol.376, Year. 2008, Page:174-9,
301.

Self Assembled Mercapto Compound-Gold-Nanoparticle Modified Carbon Paste Electrode for Potentiometric Determination of Cadmium(II)


Authors: Mashhadizadeh, MH., Eskandari, K.,Foroumadi, A., Shafiee. A
Electroanalysis, Vol.20, No.17, Year. 2008, Page:1891-6,
302.

Synthesis and in-vitro antibacterial activity of 5-substituted-1-methyl-4-nitro-1H-imidazoles


Authors: Letafat, B., Emami, S., Aliabadi, A., Mohammadhosseini, N., Moshafi, M. H., Asadipour, A., Shafiee, A., Foroumadi, A
Archiv der Pharmazie - Chemistry in Life Science, Vol.341, Year. 2008, Page:501-497,
303.

Synthesis and in vitro anti-Helicobacter pylori activity of 2-[(chlorobenzyl)thio]-5-(5-nitro-2-furyl)-1,3,4- thiadiazoles


Authors: Mohammadhosseini, N., Letafat, B., Siavoshi, F., Emami, S., Safari, F., Shafiee, A., Foroumadi, A
Med Chem Res, Vol.17, Year. 2008, Page:586-578,
304.

Structure-Activity Relationship Study of a Series of N-Substituted Piperazinyl-Fluoroquinolones as Anti-Helicobacter pylori Agents


Authors: Foroumadi, A., Safavi, M., Emami, S., Siavoshi, F., Najjari, S., Safari, F., Shafiee, A
Medicinal Chemistry, Vol.4, No.5, Year. 2008, Page:502-498,
305.

Synthesis and cytotoxic activity of novel chromenes


Authors: Alizadeh B. H., Ostad S. N., Foroumadi A., Amini M., Dowlatabadi R., Navidpour L., Shafiee A
ARKIVOK, Vol.13, Year. 2008, Page:56-45,
306.

Synthesis and in-vitro antibacterial activity of N-piperazinyl quinolone derivatives with 5-chloro-2-thienyl group


Authors: Shafiee A., Haddad Zahmatkesh M., Mohammadhosseini N., Khalafy J., Emami S., Moshafi MH., Sorkhi M., Foroumadi A
DARU , Vol.16, No.3, Year. 2008, Page:195-189,
307.

Copper(II) modified carbon paste electrodes based on self-assembled mercapto compounds-gold-nanoparticle


Authors: Mashhadizadeh, MH., Eskandari, K.,Foroumadi, A., Shafiee. A
Talanta, Vol.76, Year. 2008, Page:502-497,
308.

Enantioselective determination of tramadol and its main phase I metabolites in human plasma by high-performance liquid chromatography


Authors: Ardakani, YH., Mehvar, R., Foroumadi, A., Rouini, MR
Journal of Chromatography B, Vol.864, Year. 2008, Page:115-109,
309.

Spectrophotometric determination of acidity constants by two-rank annihilation factor analysis


Authors: Hemmateenejad, B., Abbaspour, A., Maghami, H., Foroumadi, A
Analytical Chimica Acta, Vol.607, Year. 2008, Page:152-142,
310.

Synthesis and antibacterial activity of quinolone-based compounds containing a coumarin moiety


Authors: Emami, S., Foroumadi, A., Faramarzi, MA., Samadi, N
Arch. Pharm. Chem. Life Sci, Vol.341, Year. 2008, Page:48-42,
311.

Synthesis and evaluation of antioxidant activity of novel 6-methoxy-2H-chromenes


Authors: Sorkhi, M., Forouzani, M., Dehghan, Gh., Abdollahi, M., Shafiee, A., Foroumadi, A
Asian J. Chem, Vol.20, No.3, Year. 2008, Page:2155-2151,
312.

New synthetic route towards 2,2-dimethylchromene and synthesis of substituted 7-(dimethylpropargyl) chromene


Authors: Alizadeh, B.H., Foroumadi, A., Shafiee, A
J. Heterocyclic Chem, Vol.45, Year. 2008, Page:912-909,
313.

2-Hydroxyphenacyl azoles and related azolium derivatives as antifungal agents


Authors: Emami, S., Foroumadi, A., Falahati, M., Lotfali, E., Rajabalian, S., Ebrahimi, S. A., Farahyar, S., Shafiee, A.
Bioorg. Med. Chem. Lett, Vol.18, Year. 2007, Page:146-141,
314.

Synthesis, antituberculosis activity and QSAR study of some novel 2-(nitroaryl)-5-(nitrobenzylsulfinyl and sulfonyl)-1,3,4-thiadiazoloe derivatives


Authors: Foroumadi, A., Sakhteman, A., Sharifzadeh, Z., Mohammadhosseini, N., Hemmatinejad, B., Moshafi, M. H., Vosooghi, M., Amini, M., Shafiee, A
Daru, Vol.15, No.4, Year. 2007, Page:226-218,
315.

Synthesis and antioxidant properties of substituted 3-benzylidene-7-alkoxychromsanon-4-ones


Authors: Foroumadi A., Samzadeh-Kermani, A., Emami, S., Dehghan, G., Sorkhi, M., Arabsorkhi, F., Heidari, M. R., Abdollahi, M., Shafiee, A
Bioorg. Med. Chem. Lett, Vol.17, Year. 2007, Page:6769-6764,
316.

Synthesis, Analgesic and Anti-inflammatory activity of 4-(2-phenoxyphenyl)semicarbazones


Authors: Rineh, A., Mahmoodi, N., Abdolahi, M., Foroumadi A., Sorkhi, M., Shafiee, A
Archiv der Pharmazie, Vol.340, Year. 2007, Page:415-409,
317.

Synthesis and anticonvulsant activity of novel 2-amino-5-[4-chloro-2-(chlorophenoxy)phenyl]-1,3,4-thiadazole derivatives


Authors: Foroumadi A., Sheibani, V., Sakhteman, A., Rameshk, M., Abbsi, M., Farazifard, R., Tabatabai, S.A., Shafiee, A
Daru, Vol.15, No.2, Year. 2007, Page:93-89,
318.

A mechanistic QSAR study on the leishmanicidal activity of some 5-substituted-1,3,4-thiadiazole derivatives


Authors: Hemmateenejad, B., Miri, R., Niroomand, U., Foroumadi A., Shafiee, A
Chem. Biol. Drug Des, Vol.69, Year. 2007, Page:443-435,
319.

Synthesis and antibacterial activity of levofloxacin derivatives with certain bulky residues on piperazine rings


Authors: Foroumadi A., Emami S., Mansouri, S., Javidnia, A., Saeid-Adeli, N., Shirazi, F. H., Shafiee, A
European J. Med. Chem, Vol.42, Year. 2007, Page:992-985,
320.

In vitro cytotoxicity and phototoxicity of N-piperazinyl quinolone derivatives with a 2-thienyl group


Authors: Pardakhti, A., Foroumadi A., Hashemi, M., Rajabalian, S., Heidari, M
Toxicology in vitro, Vol.21, Year. 2007, Page:1038-1031,
321.

Synthesis and antibacterial activity of new N-[2-(thiophen-3-yl)ethyl]piperazinyl quinolones


Authors: Letafat, B., Emami, S., Mohammadhosseini, N., Faramarzi, M.A., Samadi, N., Shafiee, A., Foroumadi A
Chem. Pharm. Bull, Vol.55, No.6, Year. 2007, Page:898-894,
322.

Synthesis of new fluoroquinolones containing a N-[5-(fluorobenzylthio)-1,3,4-thiadiazole-2-yl]piperazine moiety


Authors: Foroumadi A., Firoozpour, L., Nematollahi, N., Ebrahimabadi, A.H., Emami, S., Moshafi, M., Asadipour, A., Shafiee, A
Asian J. Chem, Vol.19, No.6, Year. 2007, Page:4552-4547,
323.

Theoretical study on Z/E selectivity in the oximation of α-haloacetophenones


Authors: Emami, S., Foroumadi A
Asian J. Chem, Vol.19, No.6, Year. 2007, Page:4732-4727,
324.

Synthesis of 2-alkyl-1-[4-(5-carboxy-1,2,3-thiadiazole-4-yl)benzyl]-4-chloro-1H-imidazole-5-carboxaldehydes


Authors: Amini, M., Foroumadi A., Vossghi, M., Vahdatizadeh, H., Shafiee, A
Asian J. Chem, Vol.19, No.6, Year. 2007, Page:4683-4679,
325.

Functionalized N-(2-oxyiminoethyl)piperazinyl quinolones as new cytotoxic agents


Authors: Rajabalian, S., Foroumadi A., Shafiee, A., Emami, S
J. Pharm. Pharmaceut Sci, Vol.10, No.2, Year. 2007, Page:158-153,
326.

Synthesis and antibacterial activity of N-[5-(chlorobenzylthio)-1,3,4-thiadiazol-2-yl] piperazinyl quinolone derivatives


Authors: Foroumadi A., Firoozpour, L., Emami S., Mansouri, S., Ebrahimabadi, A. H., Asadipour, A., Amini, M., Saeid-Adeli, N., Shafiee, A
Arch. Pharm. Res, Vol.30, No.2, Year. 2007, Page:145-138,
327.

Synthesis and antibacterial activity of new 7-piperazinyl-quinolones containing a functionalized 2-(furan-3-yl)ethyl


Authors: Foroumadi A., Mohammadhosseini N., Emami S., Letafat B., Faramarzi M. A., Samadi N., Shafiee A
Arch. Pharm. Chem. Life Sci, Vol.340, Year. 2007, Page:52-47,
328.

Synthesis and antioxiodant activity of some novel 2-amino-4-aryl-3-cyano-7-(dimethylamino)-4H-chromenes


Authors: Foroumadi A., Dehghan Gh., Samzadeh A., Arabsorkhi F., Sorkhi M., Shafiee A., Abdollahi M
Asian J. of Chemistry, Vol.19, No.2, Year. 2007, Page:1396-1391,
329.

Evaluation of invitro leshmanicidal activity of novel 1,3,4-thiadiazole derivatives against L.major


Authors: Nosratabadi S.J.,Farsi-Harandi M.,Foroumadi A.,Mahmoodi M.,Daneshvar H
Journal of Rafsanjan University of Medical Sciences, Vol.6, No.2, Year. 2007, Page:100-91,
330.

Synthesis and antibacterial activity of nitro arylthiadiazole- levofloxacin hybrids


Authors: Foroumadi A., Mansouri S., Emami S., Mirzaie J., Sorkhi M., Saeid-Adeli N., Shafiee A
Arch. Pharm. Chem. Life Sci, Vol.339, Year. 2006, Page:624-621,
331.

Evaluation of in vitro Antimicrobial effectiveness of novel Nitro imidazole and Nitrofurane Derivatives Against Helicobacter pylori


Authors: Foroumadi A., Siavoshi F., Safari F., Sheikholeslami A., Massarrat S
Helicobacter, Vol.11, No.4, Year. 2006, Page:398,
332.

Thrombomodulin induction in cultured human endothial cells by 9-cis-locked retinoic acid analogues


Authors: Bioorganic & Medicinal Chemistry
Ikegami S., Iimori T., Sudo M., Kitsukawa M., Foroumadi A., Yonemura T., Takahashi H., Kizaki K., Ishii H, Vol.14, Year. 2006, Page:5109-5099,
333.

Synthesis of 4-(4-methyl sulfonylphenyl)-3-phenyl-2(3H)-thiazole Thione Derivatives as Potential COX-2 Inhibitors


Authors: Emami S., Foroumadi A
Chinese J. Chemistry, Vol.24, No.6, Year. 2006, Page:794-791,
334.

Synthesis and Anti bacterial activity of new fluoroquinolones containing a substituted N-(phenethyl)piperazine moiety


Authors: Foroumadi A., Ghodsi S., Emami S., Najjari A., Samadi N., Faramarzi M.A., Beikmohammadi L., Shirazi F.H., Shafiee A
Bioorganic & Medicinal Chemistry Letters, Vol.16, Year. 2006, Page:3503-3499,
335.

Synthesis and antibacterial activity of N-[2-[5-(methylthio)thiophen-2-yl]-2-oxoethyl] and N-[2-[5-(methylthio)thio phen-2-yl]-2-(oxyimino)ethyl]piperazinylquinolone derivatives


Authors: Foroumadi A., Oboudiat M., Emami S., Karimollah A., Saghaee L., Moshafi M. H., Shafiee A
Bioorg. Med. Chem, Vol.14, Year. 2006, Page:3421-7,
336.

Structural Feature of New Quinolones and Relationship to Antibacterial Activity against Gram-Positive Bacteria


Authors: Emami S., Shafiee A., Foroumadi A
Mini- Reviews in Medicinal Chemistry, Vol.6, Year. 2006, Page:386-375,
337.

A Rapid and Sensitive HPLC Method for the Determination of 2-hydroxyflutamide in Human Plasma


Authors: Jalalizadeh H., Souri E., Javadi Ghanami H.R., Almasirad A., Foroumadi A
International Journal of Pharmacology, Vol.2, No.2, Year. 2006, Page:225-221,
338.

Synthesis and antimicobacterial activity of some alkyl [5-(nitroaryl)-1, 3, 4- thiadiazol-2-ylthio]propionates


Authors: Foroumadi A., Kargar Z., Sakhteman A., Sharifzadeh Z., Feyzmohammadi R., Kazemi M., Shafiee A
Bioorg. Med. Chem. Lett, Vol.16, Year. 2006, Page:1167-1164,
339.

Development and validation of a rapid HPLC method for simultaneous determination of tramadol, and its two main metabolites in human plasma


Authors: Rouini M., Hoseinzadeh Ardakani Y., Soltani F., Aboul-Enein H., Foroumadi A
J. Chromatogr. B Analyt. Technol. Biomed. Life Sci, Vol.830, Year. 2006, Page: 211-207,
341.

Synthesis and in vitro leishmanicidal activity of 2-(1-methyl-5-nitro-1H-imidazol-2-yl)-5-substituted- 1,3,4-thiadiazole derivatives.


Authors: Foroumadi A., Emami S., Pournourmohammadi S., Kharazmi A., Shafiee A
Eur. J. Med. Chem, Vol.40, Year. 2005, Page:1350-1346,
342.

Synthesis and antibacterial activity of N-[2-(5-bromothiophen-2-yl)-2-oxoethyl] and N-[(2-(5-bromo thiophen-2-yl)-2-Oximinoethyl] derivatives of piperazinyl quinolones


Authors: Foroumadi A., Emami S., Mehni M., Moshafi M., Shafiee A
Bioorg. Med. Chem. Lett, Vol.15, Year. 2005, Page:4539-4536,
343.

Synthesis and antibacterial activity of N-(5-benzylthio-1,3,4- thia diazol-2-yl) piperazinyl quinolone derivatives.


Authors: Foroumadi A., Emami S., Hassanzadeh A., Rajaee M., Sokhanvar K.,Moshafi M., Shafiee A
Bioorg. Med Chem. Lett, Vol.15, Year. 2005, Page:4492-4488,
344.

Syntheses of N-[3-(1-methyl-1H-2-imidazolyl) propyl] benzamides and N-[3-(1-­methyl-lH-2-imidazolyl)propyl] benzenesulfon amides


Authors: Shafiee A., Shabani P., Vosooghi M., Foroumadi A
J. Heterocyclic Chem, Vol.42, Year. 2005, Page:1015-1011,
345.

Synthesis and in vitro leishmanicidal activity of 2-(5-nitro-2-furyl) and 2-(5-nitro-2-thienyl)-5- substituted­-1,3,4-thiadiazoles.


Authors: Foroumadi A., Pournourmohammadi S., Soltani F., Asgharian Rezaee M., Dabiri S., Kharazmi A., Shafiee A
Bioorg. Med Chem. Lett, Vol.15, Year. 2005, Page:1985-1983,
346.

Synthesis, in vitro-Antimycobacterial Activity and Cytotoxicity of Some Alkyl α-(5-aryl-1,3,4-thiadi­azole-2-ylthio)acetates,.


Authors: Foroumadi A., Soltani F., Moallemzadeh-Haghighia H., Shafiee A
Arch Pharm Chem. Life Sci, Vol.338, Year. 2005, Page:116-112,
347.

Synthesis And Conversion of Ethyl 4-(4-Methyl phenyl)-1,2,3-Selenadiazole-5-Carboxylate To Ethyl 3-(4-Methylphenyl) Propiolate


Authors: Foroumadi A., Amini M., Vosooghi M., Vahdatizade H., Shafiee A
Chem. Ind. J, Vol.1, No.11, Year. 2005, Page:709-707,
348.

Synthesis and Antifungal Evaluation of Allyl Containing Derivatives Of 5-(5-Nitrofuran-2-yl)-1,3,4-Thiadiazole


Authors: Emami S., Foroumadi A
Chem. Ind. J, Vol.2, No.1, Year. 2005, Page:13-10,
349.

Synthesis Of Methyl 1,4-Dihydro-2,6-Dimethyl-3-Nitro-4-(4,5-Dichloro imidazol-2-yl)-5-Pyridine Carboxylate as Potential Calcium Channel Modulator


Authors: Foroumadi A., Bakhtiari D., Amini M., Shafiee A
Chem. Ind. J, Vol.2, No.1, Year. 2005, Page:9-7,
350.

Quinoloines: Recent Structureal and Clinical Developments


Authors: Emami S., Shafiee A., Foroumadi A
Iranian J. Pharm. Res, Vol.3, Year. 2005, Page:136-123,
351.

Synthesis Of 1-(Furan-2-yl)-2-(1H-Imidazol-1-yl) Ethanone O-Benzyloxime As A Furan Analog Of Oxiconazole


Authors: Emami S., Foroumadi A., Asadipour A., Toyserkani A
Chem. Ind. J, Vol.1, No.12, Year. 2005, Page:751-749,
352.

Chemical Composition Of The Essential Oil Of Satureja hortensis L. var.laxiflora


Authors: Foroumadi A., Asadipour A., Maddah B., Senemar S., Mehrabani M
Chem. Ind. J, Vol.1, No.10, Year. 2005, Page:702-701,
353.

Synthesis Of Certain Diarylsulfonylurea Derivatives As New Potential Antitumor Agents


Authors: Foroumadi A., Emami S., Rezvani N., Shafiee A., Asadipour A
Chem. Ind. J, Vol.1, No.12, Year. 2005, Page:748-745,
355.

Synthesis and in vitro antibacterial evaluation of N-[5-(5-nitro-2-thienyl)-1, 3, 4-thiadiazole-2-yl] piperazinyl quinolones


Authors: Foroumadi A., Mansouri S., Kiani Z., Rahmani A
Eur. J. Med. Chem, Vol.38, No.9, Year. 2003, Page:851-4,
356.

Synthesis and in vitro antibacterial activity of some N-(5-aryl-1,3,4-thiadiazole-2-yl) piperazinyl quinolone derivatives


Authors: Foroumadi A., Soltani F., Moshafi M., Ashraf-Askari R
IlFarmaco, Vol.58, No.10, Year. 2003, Page:1023-8,
359.

Antituberculosis agents. VII. Synthesis and in vitro evaluation of antimycobacterial activity and cytotoxicity of some N-piperazinyl quinolone derivatives


Authors: Foroumadi A., Soltani F., Asadipour A
Boll. Chim. Farm, Vol.142, No.3, Year. 2003, Page:130-4,
360.

Synthesis and in vitro antibacterial activity of N-[5-(5-nitro-2-furyl)-1,3,4-thiadiazole-2-yl] piperazinyl quinolone derivatives


Authors: Foroumadi A., Ashraf-Askari R., Moshafi M., Emami S., Zeynali A
Pharmazie, Vol.58, No.6, Year. 2003, Page:432-3,
361.

Synthesis and evaluation of in vitro antimycobacterial activity of some 5-(5-nitro-2-thienyl)-2-(piperazinyl, piperidinyl and morpholinyl)-1,3,4-thiadiazole derivatives


Authors: Foroumadi A., Soltani F., Rezaee M., Moshafi M
Boll. Chim.Farm, Vol.142, No.9, Year. 2003, Page:416-9,
362.

Anti – pseudomona and anti – bacilli activity of some medicinal plant of Iran


Authors: Shadidi Bonjar G., Karimi Nik A., Heydari M., Ghasemzadeh M., Farrokhi P., Moein M., Mansouri S., Foroumadi A
Daru , Vol.11, No.4, Year. 2003, Page:163-157,
364.

Composition of the essential oil of Bunium persicum B. Fedthech from Iran


Authors: Foroumadi A., Asadipour A., Amanzadeh Y., Arabpour F
J. Essential Oil Res, Vol.14, Year. 2002, Page:162-161,
365.

Antituberculosis agents. III. In vitro evaluation of anti mycobacterial activity and cytotoxicity of some N- piperaziny quinolone derivatives


Authors: Foroumadi A., Soltani F., Emami S., Davood A
Boll. Chim. Farm, Vol.141, No.3, Year. 2002, Page:247-9,
366.

Cytotoxic activity of medicinal plants used in Iranian traditional medicine on two strains of saccharomyces cervisiae


Authors: Shahidi Gh., Moein M., Foroumadi A., Rokhbakhsh – Zamin F
Daru, Vol.10, No.4, Year. 2002, Page:164-162,
367.

Synthesis and calcium channel antagonist activity of nifedipine analogues with methylthiomidazole substituent


Authors: Foroumadi A., Analuie N., Rezvanipour M., Sepehri G., Najafipour H., Sepehri H., Javanmardi K., Esmaeeli F
IL Farmaco, Vol.57, Year. 2002, Page:199-195,
368.

Synthesis and in vitro antimicrobial evaluation of 5-(1-methyl-5-nitro-2-imidazolyl)-4H-1,2,4-triazoles


Authors: Shafiee A., Sayadi A., Roozbahani M., Foroumadi A., Kamal F
Arch. Pharm. (Weinheim) , Vol.335, No.10, Year. 2002, Page:495-9,
369.

Activity of a new ciprofloxacin derivative against Mycobacterium avium and some drug-resistant strains of Mycobacterium tuberculosis


Authors: Foroumadi A., Soltani F., Moshafi M. Antituberculosis agents. VI
Boll. Chim. Farm, Vol.141, No.5, Year. 2002, Page:394-6,
370.

Synthesis, evaluation of in vitro antituberculosis activity and cytotoxicity of some 2-(5-nitro-2-furyl)-1, 3, 4-thiadiazole derivatives


Authors: Foroumadi A., Asadipour A., Mirzaei M., Karimi J., Emami S. Anti tuberculosis agents. V
Farmaco, Vol.57, No.9, Year. 2002, Page:765-9,
371.

Synthesis and Antifungal Activity of some New 1,2,4- Triazole [3,4-a] thiadiazine derivatives


Authors: Foroumadi A., Mirzaei M., Emami S., Salari P., Ghaffari F., Amini M., Shafiee A
Daru, Vol.10, No.1, Year. 2002, Page:37-34,
372.

Synthesis and evaluation of antibacterial activity of some novel N-substituted piperazinyl quinolones


Authors: Foroumadi A., Davood A., Mirzaei M., Emami S., Moshafi M
Boll. Chim. Farm, Vol.140, Year. 2001, Page:416-411,
373.

Antibacterial activity of the crude extracts and frctionated constituents of Myrtus communis


Authors: Mansouri S., Foroumadi A., Ghaneie T., Gholamhoseinian Najar A
Pharmaceutical Biology, Vol.39, Year. 2001, Page:401-399,
375.

Antituberculosis Agents I. Synthesis and Antituberculosis Activity of 2-Aryl-1,3,4-thiadiazole Derivatives


Authors: Foroumadi A., Mirzaei M., Shafiee A
Pharmazie, Vol.56, Year. 2001, Page:612-610,
376.

Synthesis and in-vitro antibacterial activities of N-piperazinyl quinolone derivatives with 2-thienyl group


Authors: Mirzaei M., Foroumadi A
Pharm. Pharmacol. Commun, Vol.6, Year. 2000, Page:351-35,
377.

Synthesis and Anticonvulsant Activity of 5-Aryl-1, 3, 4- thiadiazole Derivatives


Authors: Foroumadi A., Tabatabaie A., Gitnezhad G., Zarrendast M., Shafiee A
Pharm. Pharmacol. Commun, Vol.6, Year. 2000, Page:33-31,
378.

Synthesis and anti-inflamatory activity of 1-methyl-5- (4-X-benzoyl) imidazole-2- acetates


Authors: Shafiee A., Kaabinejadian S., Foroumadi A., Zarrindast M
Pharm. Pharmaco. Commun, Vol.5, Year. 1999, Page:275-273,
379.

Synthesis and in vitro anti fungal activity of 2-aryl-5-phenylsufonyl-1,3,4-thiadiazole derivatives


Authors: Foroumadi A., Daneshtalab M., Shafiee A
Arzeneimittel Forschung Drug Research, Vol.49, Year. 1999, Page:1038-1035,
380.

Synthesis and in-vitro antibacterial activity of new N-substituted piperazinyl quinolones


Authors: Foroumadi A., Emami S., Haghighat P., Moshafi M
Pharm. Pharmacol. Commun, Vol.5, Year. 1999, Page:594-591,
381.

Syntheses and antifungal activity of 2-aryl -1,3,4- thiadiazole 5-fulfide, sulfoxide and sulfones


Authors: Foroumadi A., Daneshtalab M., Mahmoudian M., Falahati M.,Nateghian N., Shahsavarani N., Shafiee A.
Pharm. Pharmacol Commun, Vol.4, Year. 1998, Page:98-95,
382.

Syntheses of 2-(2-Arylethyl) imidazoles


Authors: Shafiee A., Rastkary N., Foroumadi A
J. Heterocyclic Chem, Vol.35, No.3, Year. 1998, Page:610-607,
383.

Syntheses of 4 and 5-Alkylsulfonylimidazoles


Authors: Shafiee A., Akbarzadeh T., Foroumadi A., Hadizadeh F
J. Heterocyclic Chem, Vol.35, No.1, Year. 1998, Page:144-141,
384.

Syntheses and In vitro antibacterial activities of N-Substituted piperazinyl quinolones


Authors: Foroumadi A., Emami A., Davood A., Moshafi M., Sharifian A., Tabatabaie M., Tarhimifarimani H., Sepehri G., Shafiee A
Pharm. Sciences, Vol.3, Year. 1997, Page:563-559,
385.

Syntheses of substituted pyrrolo [3,2-d] imidazoles


Authors: Shafiee A., Hadizadeh F., Foroumadi A
Ind. J. Chem. (Sec.B), Vol.36, No.9, Year. 1997, Page:815-813,
386.

Synthesis of 2-(2-Aryl ethyl)-1- methylimidazoles


Authors: Shafiee A., Morteza-semnani K., Foroumadi A
J. Heterocyclic Chem, Vol.33, No.3, Year. 1996, Page:673-671,
387.

Synthesis of Arylsulfonyl -1,3,4- thiadiazoles


Authors: Shafiee A., Foroumadi A
J. Heterocyclic Chem, Vol.33, No.6, Year. 1996, Page:1614-1611,
388.

Syntheses of substituted Oxazolo –1,3,4-thiadiazoles, 1,3,4- oxadiazolers and 1,2,4-triazoles


Authors: Shafiee A., Naimi E., Mansobi P., Foroumadi A., Shekari M
J. Heterocyclic Chem, Vol.32, No.4, Year. 1995, Page:1239-1235,
389.

Syntheses of substituted (1,3,4-oxadiazole-2-yl)-4- nitropyrroles and 1-Methyl 4-nitropyrrole-2- (1, 3, 4-thiadiazole -2-yl-4-nitropyrroles


Authors: Firoozi F., Javidnia K., Kamali M., Fooladi A., Foroumadi A., Shafiee A
J. Heterocyclic Chem, Vol.32, No.1, Year. 1995, Page:128-123,
390.

Synthesis of 1,3,4-thiadiazoles and 1,3,4-oxadiazoles: 2-(1-Methyl-4-nitro-2-pyrroly) –5- substituted –1,3,4-thiadiazoles and 1,3,4-oxadiazoles


Authors: Shafiee A., Firoozi F., Javidnia K., Kamali M., Fooladi A., Foroumadi A
Phosphorus Sulfur and Silicon, Vol.96-95, Year. 1994, Page:472-471,

Farsi

1.

Editorial Board of Iranian Journal of Pharmaceutical Research


Activity Type:Member
1. Screening of the medicinal plants for Anti - Helicobacter pylori activity
2. Synthesis of new potent anti-Helicobacter pylori agents
3. Synthesis of new potent anti - leishmania agents
4. Synthesis of rigid Retinoic acid derivatives (for use as anticancer agents) and other biologically active compounds using modern
5. Synthesis of potent cytotoxic agents from fluoroquinolone series for use as anticanser agents
6. The major objective of my research program in medicinal Chemistry Concerns the design, synthesis and biological evaluation of an
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